Target Details
| UniProt AC | Q6DT37 |
|---|---|
| Gene Symbol | CDC42BPG |
| Protein Name | Serine/threonine-protein kinase MRCK gamma |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00780 (CNH) PF08826 (DMPK_coil) PF25346 (PH_MRCK) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 13
- Clinical molecules 4
- Avg pChEMBL 6.96
Active Molecules (13)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.1 | IC50 | 408 | — | |
NXSJMRCTGYTSTK
|
8.2 | Kd | 200 | — | |
HKSZLNNOFSGOKW
|
7.4 | Kd | 213 | — | |
DKZYXHCYPUVGAF
|
7.2 | Kd | 112 | — | |
MWKSRKSEWLRPBL
|
7.0 | Kd | 1075 | — | |
CXQHYVUVSFXTMY
|
6.8 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.7 | Kd | 149 | — | |
VAARYSWULJUGST
|
6.6 | Kd | 119 | Yes | |
PBCZSGKMGDDXIJ
|
6.6 | Kd | 68 | Yes | |
CDMGBJANTYXAIV
|
6.4 | Kd | 34 | Yes | |
BPNUQXPIQBZCMR
|
6.3 | Kd | 83 | Yes | |
QHKYPYXTTXKZST
|
6.2 | Kd | 28 | — | |
QVOGVAVHOLLLAZ
|
6.1 | Kd | 4 | — |