Target Details
| UniProt AC | Q5VT25 |
|---|---|
| Gene Symbol | CDC42BPA |
| Protein Name | Serine/threonine-protein kinase MRCK alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00780 (CNH) PF08826 (DMPK_coil) PF15796 (KELK) PF25346 (PH_MRCK) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 233
- Clinical molecules 60
- Avg pChEMBL 7.87
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CFIBXVQLBVNOHW
|
6.0 | Ki | 64 | — | |
HTROFVQKJODSCL
|
6.0 | Ki | 11 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NGFGTMFVWSDFPS
|
6.0 | IC50 | 32 | — | |
UUWNXFJBBYAMDT
|
6.0 | Ki | 46 | — | |
XMFUGSRATNLPRM
|
6.0 | Ki | 19 | — | |
ZRTWUBWXIGHVET
|
6.0 | Ki | 10 | — | |
AAAXBDFZRXKRPL
|
Clinical | TTD_MultiTarget | 6 | Yes | |
APMQKHHNTLVDQD
|
Clinical | TTD_MultiTarget | 6 | Yes | |
AWPVKERKWQLOEG
|
Clinical | TTD_MultiTarget | 4 | Yes | |
BPGIPYJOESFNQI
|
Clinical | TTD_MultiTarget | 6 | Yes | |
CCUWZTRFTGLQCV
|
Clinical | TTD_MultiTarget | 5 | Yes | |
CLYHSTKBWHUKBD
|
Clinical | TTD_MultiTarget | 2 | Yes | |
GLDPXWNDIUPOHH
|
Clinical | TTD_MultiTarget | 6 | Yes | |
HDJINRKHYZJXSV
|
Clinical | TTD_MultiTarget | 3 | Yes | |
HKNVXYDHMZZSGS
|
Clinical | TTD_MultiTarget | 3 | Yes | |
HTUPONJUVMCVCW
|
Clinical | TTD_MultiTarget | 6 | Yes | |
INASOKQDNHHMRE
|
Clinical | TTD_MultiTarget | 2 | Yes | |
KKVYYGGCHJGEFJ
|
Clinical | TTD_MultiTarget | 6 | Yes | |
MEQSMKIFBMBPQX
|
Clinical | TTD_MultiTarget | 6 | Yes | |
MHVFDATVTOZXQW
|
Clinical | TTD_MultiTarget | 6 | Yes | |
MLDQJTXFUGDVEO
|
Clinical | TTD_MultiTarget | 85 | Yes | |
MRKUZTPMEBRBGD
|
Clinical | TTD_MultiTarget | 6 | Yes | |
OYAMULIHRWEUAR
|
Clinical | TTD_MultiTarget | 7 | Yes | |
QLKGZBYGKCVLEX
|
Clinical | TTD_MultiTarget | 5 | Yes | |
UPABYWZSQBEEII
|
Clinical | TTD_MultiTarget | 6 | Yes | |
UTVABCSMEKUFLJ
|
Clinical | TTD_MultiTarget | 7 | Yes | |
VVYFYJMXONNWBA
|
Clinical | TTD_MultiTarget | 7 | Yes | |
YEUIDIRYOPOAPU
|
Clinical | TTD_MultiTarget | 5 | Yes | |
YLQMVIRZBOJBCV
|
Clinical | TTD_MultiTarget | 7 | Yes | |
ZJZMAUBKRKIVPH
|
Clinical | TTD_MultiTarget | 3 | Yes |