Target Details
| UniProt AC | Q5VT25 |
|---|---|
| Gene Symbol | CDC42BPA |
| Protein Name | Serine/threonine-protein kinase MRCK alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00780 (CNH) PF08826 (DMPK_coil) PF15796 (KELK) PF25346 (PH_MRCK) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 233
- Clinical molecules 60
- Avg pChEMBL 7.87
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OLUKILHGKRVDCT
|
6.7 | Ki | 44 | Yes | |
SOVYWBOZOBVFLP
|
6.7 | Ki | 10 | — | |
XSDJOIOVIMPMHD
|
6.7 | Ki | 44 | — | |
ZRQXCQXWTLVASO
|
6.7 | Ki | 36 | — | |
DNAXPHDUUNPFLH
|
6.7 | IC50 | 2 | — | |
VIKNJXKGJWUCNN
|
6.6 | pIC50 | 6 | Yes | |
OMVMGDVRMSCTFN
|
6.6 | IC50 | 3 | — | |
AOBLBPWPSKBHSI
|
6.6 | Ki | 55 | — | |
CLRFYTGANQZOBS
|
6.6 | Ki | 41 | — | |
JCTPJYZESAMIGH
|
6.6 | Ki | 2 | — | |
JXMYIDZREHNPDO
|
6.6 | Ki | 19 | — | |
WNMXOXGXHRHBLO
|
6.6 | Ki | 4 | — | |
PBCZSGKMGDDXIJ
|
6.6 | Kd | 68 | Yes | |
KGVGNTCIQIYLQU
|
6.5 | pIC50 | 9 | Yes | |
BSFNGHCTZDCQBF
|
6.5 | Ki | 93 | — | |
MLGGUGPIWDHBAI
|
6.5 | Ki | 33 | — | |
RFVBRKXQYUDGIO
|
6.5 | Ki | 23 | — | |
USHMNZBDAOGLMB
|
6.5 | Ki | 26 | — | |
VGNKOJURPOHWJF
|
6.5 | Ki | 21 | — | |
BKCNFBWOOAHROL
|
6.5 | IC50 | 3 | — | |
VGRBFVDNFGSMNW
|
6.4 | IC50 | 3 | — | |
BPNUQXPIQBZCMR
|
6.4 | Kd | 83 | Yes | |
LXMSZDCAJNLERA
|
6.4 | pIC50 | 6 | Yes | |
PFCUZXCHLYIMTJ
|
6.4 | Ki | 18 | — | |
DPRGOXVMSNDADU
|
6.3 | Ki | 16 | — | |
GVMDVMPNOAVKJR
|
6.3 | Ki | 26 | Yes | |
KYACBMRLQMEIAI
|
6.3 | Ki | 30 | — | |
XYZNKCSDQRKAFR
|
6.3 | Ki | 53 | — | |
ASUGUQWIHMTFJL
|
6.2 | Kd | 18 | — | |
AWJPVXSHMIELNJ
|
6.2 | Ki | 23 | — | |
BIIVYFLTOXDAOV
|
6.2 | Ki | 31 | — | |
IQNOGQGSOHNMCL
|
6.2 | Ki | 14 | — | |
LRZYYIZFBXFSJB
|
6.2 | Ki | 69 | — | |
NMWSFHOBJVDICZ
|
6.2 | Ki | 2 | — | |
NTCBYBDADUSXSB
|
6.2 | pIC50 | 9 | Yes | |
SRUYMJRFVGLQDV
|
6.2 | Ki | 37 | — | |
ZYTFPHRVOZXPGZ
|
6.2 | Ki | 30 | — | |
CXQHYVUVSFXTMY
|
6.2 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.2 | Kd | 149 | — | |
GFWDPXHTWJXOEI
|
6.2 | IC50 | 3 | — | |
KVPALVACWJUWHG
|
6.1 | pIC50 | 6 | Yes | |
FLEAYYMORDPWAJ
|
6.1 | Ki | 90 | — | |
OPOGDZANLATWGS
|
6.1 | Ki | 9 | — | |
PCQMERRARZKTPW
|
6.1 | Ki | 68 | — | |
QEWSTOOMTBAUAG
|
6.1 | Ki | 17 | — | |
QUZYEJUYJAWLOF
|
6.1 | Ki | 4 | — | |
ZPVLRSVLOWVDJC
|
6.1 | Ki | 14 | — | |
ZNDQOACBIHODQO
|
6.1 | IC50 | 3 | — | |
PSGAAPLEWMOORI
|
6.0 | pIC50 | 11 | Yes | |
PSGAAPLEWMOORI
|
6.0 | pIC50 | 3 | Yes |