Target Details
| UniProt AC | Q5VT25 |
|---|---|
| Gene Symbol | CDC42BPA |
| Protein Name | Serine/threonine-protein kinase MRCK alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00780 (CNH) PF08826 (DMPK_coil) PF15796 (KELK) PF25346 (PH_MRCK) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 233
- Clinical molecules 60
- Avg pChEMBL 7.87
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XWQDAOOPQZIBIA
|
7.7 | Ki | 4 | — | |
OUJZYQBEFNDJQN
|
7.7 | Ki | 71 | — | |
YXKBVHXOKVRRKO
|
7.7 | pIC50 | 6 | Yes | |
WFESRNFSHAPECN
|
7.7 | pIC50 | 4 | Yes | |
GHPFQRTVUDXWCC
|
7.6 | Ki | 35 | — | |
OSVUGUHRKMMBSE
|
7.6 | Kd | 170 | — | |
UAQJVFADAYIBGC
|
7.6 | Ki | 23 | — | |
LIZZRPJKAHJFGK
|
7.5 | Ki | 2 | — | |
MWKSRKSEWLRPBL
|
7.5 | Kd | 1075 | — | |
FUMCKNCUEAQHCV
|
7.5 | Ki | 103 | — | |
UPPGGRZNGRFDAU
|
7.5 | Ki | 21 | — | |
XOMYQWBAFPYLRJ
|
7.5 | Ki | 3 | — | |
ZDCMJDVSSLHLLQ
|
7.5 | pIC50 | 9 | Yes | |
MASJMHFQMYAPJR
|
7.4 | Ki | 41 | — | |
VXYDJXMHISGSDA
|
7.4 | Ki | 59 | — | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — | |
ADGQNANENRDMEA
|
7.3 | Ki | 4 | — | |
KCKXYZOBGBJZEG
|
7.3 | Ki | 36 | — | |
YWTBGJGMTBHQTM
|
7.3 | Ki | 65 | — | |
ZSMCHXGGQCKXMY
|
7.3 | pIC50 | 5 | Yes | |
HKSZLNNOFSGOKW
|
7.2 | Kd | 213 | — | |
DZCWNAMURCVSNJ
|
7.2 | Ki | 4 | — | |
GPKQGYSDQQIJLW
|
7.2 | Ki | 19 | — | |
XPHWIERLJBFPFV
|
7.2 | Ki | 69 | — | |
LYADGAGFYYXXIO
|
7.1 | IC50 | 82 | — | |
RFZAHUIHPLZLLA
|
7.1 | pIC50 | 9 | Yes | |
BPNUQXPIQBZCMR
|
7.1 | Ki | 60 | — | |
GQHMZZXJWGPHDA
|
7.1 | Ki | 20 | — | |
LCKDESRGCHSHHO
|
7.1 | Ki | 18 | — | |
NRSGWEVTVGZDFC
|
7.1 | Ki | 50 | — | |
XSRHBCYNCKAFKS
|
7.1 | Ki | 45 | — | |
QUEIBWXZNMHZJD
|
7.1 | Ki | 4 | — | |
IMTGEDOKMRCXLE
|
7.0 | pIC50 | 6 | Yes | |
LOCWELCIOZHZHE
|
7.0 | Ki | 11 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
SHENEEFOURUIBP
|
7.0 | Ki | 29 | — | |
WGYAMRMJVUNILQ
|
7.0 | Ki | 3 | — | |
JDIAOFCAAPMAGG
|
6.9 | Ki | 4 | — | |
CLEGDJQQHUTCOW
|
6.9 | Ki | 43 | — | |
NEWAULHLLUCDPD
|
6.9 | Ki | 27 | — | |
VHZNRUKXHPDXMR
|
6.9 | Ki | 4 | — | |
ROFMCPHQNWGXGE
|
6.8 | IC50 | 3 | — | |
ASNQMAVHHGGQRB
|
6.8 | Ki | 14 | — | |
FDBPGAHVEGEARY
|
6.8 | Ki | 19 | — | |
YOVNFNXUCOWYSG
|
6.8 | Ki | 33 | Yes | |
ZMNWFTYYYCSSTF
|
6.8 | Ki | 18 | — | |
DYSRECIVMDGUQU
|
6.7 | Ki | 29 | — | |
GWJHMRBQEUHFOC
|
6.7 | Ki | 42 | — | |
MIYRKQLKDQNUKZ
|
6.7 | Ki | 23 | — | |
NKGLJTITEFZKAN
|
6.7 | Ki | 35 | — |