Target Details
| UniProt AC | Q5VT25 |
|---|---|
| Gene Symbol | CDC42BPA |
| Protein Name | Serine/threonine-protein kinase MRCK alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00780 (CNH) PF08826 (DMPK_coil) PF15796 (KELK) PF25346 (PH_MRCK) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 233
- Clinical molecules 60
- Avg pChEMBL 7.87
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MYDJWFCWWHPKCH
|
9.2 | pIC50 | 6 | Yes | |
BDYFDDGUXXUNJN
|
9.1 | pIC50 | 5 | Yes | |
IAUDUYJHOKBQLW
|
9.0 | pIC50 | 6 | Yes | |
PAUQSWLMXQWBGH
|
9.0 | Ki | 4 | — | |
VWFVTEZXZVPVIK
|
9.0 | Ki | 3 | — | |
YPUGASLTKIAOPT
|
9.0 | pIC50 | 6 | Yes | |
HEGUJMRUCIWLNE
|
8.9 | Ki | 4 | — | |
MMQYPFTZXJAWGY
|
8.9 | pIC50 | 5 | Yes | |
VGFSVAVGJHPQJX
|
8.9 | Ki | 3 | — | |
DITGKHUFOCLVJI
|
8.9 | Ki | 2 | — | |
KCVAVMXQQQXOLI
|
8.8 | pIC50 | 6 | Yes | |
LVCVMYKRVFAVCM
|
8.8 | pIC50 | 6 | Yes | |
DZATYSMEKYVDKI
|
8.8 | pIC50 | 6 | Yes | |
LMNVPKCUVZQIRI
|
8.7 | Ki | 2 | — | |
NTYALJAURYTROE
|
8.7 | pIC50 | 6 | Yes | |
CGDPUQIHRJHZKR
|
8.7 | Ki | 4 | — | |
NTXRXSSTKKNELF
|
8.6 | pIC50 | 5 | Yes | |
VTSLKIKDRBEGHX
|
8.6 | Ki | 4 | — | |
CTCHAYJBEBAVDT
|
8.6 | pIC50 | 6 | Yes | |
GDVRVPIXWXOKQO
|
8.5 | IC50 | 10 | — | |
UELSMLDRSQFVHG
|
8.5 | Ki | 3 | — | |
CGAGHKVPUASFJA
|
8.5 | Ki | 3 | — | |
GAUXDXUKQPFNPK
|
8.5 | pIC50 | 6 | Yes | |
VKUWSTCDZXVNIT
|
8.5 | Ki | 4 | — | |
HKSZLNNOFSGOKW
|
8.4 | Ki | 118 | — | |
MRRXULDDEFCYAJ
|
8.3 | Ki | 4 | — | |
BFSFWCMZFSXSOK
|
8.3 | Ki | 4 | — | |
JDIAOFCAAPMAGG
|
8.3 | Ki | 4 | — | |
OYQVOOXYSCKLME
|
8.3 | Ki | 4 | — | |
QIOYFTZXBUZDSU
|
8.3 | Ki | 4 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
MPRCGDPYKHWYQP
|
8.2 | Ki | 3 | — | |
PUIKISPVMMUIMT
|
8.2 | Ki | 4 | — | |
CHTMRWQLNNRRFJ
|
8.1 | Ki | 70 | — | |
NJPWCTYVEJIQBM
|
8.1 | Ki | 72 | — | |
YDNXKPCILIWEGN
|
8.1 | Ki | 3 | — | |
DXZAHRFNIIHHLC
|
8.1 | Ki | 4 | — | |
SHMZVLGXEVPHCQ
|
8.0 | Ki | 4 | — | |
IPEXHQGMTHOKQV
|
8.0 | Kd | 12 | — | |
DSQFKUKVDCXORL
|
8.0 | Kd | 4 | — | |
DLXBCJBMEVKPIX
|
8.0 | pIC50 | 9 | Yes | |
GBPXRWHRMNNALK
|
7.9 | Ki | 3 | — | |
NVVLAIWWHAUHCF
|
7.9 | Ki | 4 | — | |
KTDHNPKPSLZNRH
|
7.9 | Ki | 4 | — | |
RCADYZZSAWVHPR
|
7.8 | Ki | 4 | — | |
FNAPEKSJRDLQRC
|
7.8 | Ki | 4 | — | |
XFWUTMHVDGPWLH
|
7.8 | Ki | 75 | — | |
ZILLQAUSVGQYOB
|
7.8 | Ki | 4 | — | |
MUWPCRFJUPJCRM
|
7.7 | Ki | 4 | — | |
FJHBZDZOSWVMSE
|
7.7 | Ki | 4 | — |