Target Details
| UniProt AC | Q5TCY1 |
|---|---|
| Gene Symbol | TTBK1 |
| Protein Name | Tau-tubulin kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 12
- Clinical molecules 1
- Avg pChEMBL 7.07
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPJVZSVEIGCFJP
|
8.8 | IC50 | 2 | — | |
ISYRCGISNANONJ
|
8.0 | IC50 | 3 | — | |
DBMRETDBROLHGL
|
7.7 | IC50 | 2 | — | |
HPJVZSVEIGCFJP
|
7.5 | IC50 | 2 | — | |
WZLQQYUWMGFXDE
|
7.2 | IC50 | 3 | — | |
OPHQVUNMCJRXJP
|
6.9 | IC50 | 2 | — | |
DGLFSNZWRYADFC
|
6.7 | IC50 | 12 | — | |
BNDYIYYKEIXHNK
|
6.6 | Kd | 7 | Yes | |
QZBWRRCYSQGONG
|
6.4 | IC50 | 2 | — | |
NHZNMMAEOYALKY
|
6.4 | IC50 | 2 | — | |
BDYNACMDWPBSRV
|
6.4 | IC50 | 2 | — | |
GSVSRJBZRJBGOQ
|
6.1 | IC50 | 2 | — |