Target Details
| UniProt AC | Q5S007 |
|---|---|
| Gene Symbol | LRRK2 |
| Protein Name | Leucine-rich repeat serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23745 (ANK_LRRK2) PF23744 (ARM_LRRK2) PF23748 (Beta-prop_LRRK2) PF16095 (COR-A) PF25497 (COR-B) PF13855 (LRR_8) PF00069 (Pkinase) PF08477 (Roc) |
Summary
- Multi-target molecules 299
- Clinical molecules 21
- Avg pChEMBL 7.24
KEGG Pathways (2)
Associated Diseases (3)
Active Molecules (299)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MUCCEFIYUNZMOE
|
6.3 | IC50 | 2 | — | |
OUVFQPVWKVFPGM
|
6.3 | IC50 | 2 | — | |
SHGQVDUEFPICQD
|
6.3 | IC50 | 2 | — | |
UJLAWZDWDVHWOW
|
6.3 | Kd | 16 | — | |
VIQMKNOGQPLVRW
|
6.3 | IC50 | 2 | — | |
VONCWACGTNICLZ
|
6.3 | IC50 | 2 | — | |
VYRBWRJZNBEDCB
|
6.3 | IC50 | 2 | — | |
WJEAROLZOUZMPP
|
6.3 | IC50 | 2 | — | |
WRXKCNIVRTVEQV
|
6.3 | IC50 | 2 | — | |
YJTUMWSGGUZEFI
|
6.3 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
6.2 | IC50 | 92 | — | |
BQYDGSNDLAZAEW
|
6.2 | Ki | 13 | — | |
GCIKSSRWRFVXBI
|
6.2 | Ki | 109 | Yes | |
PHWHNHYZZNJPLB
|
6.2 | Ki | 16 | — | |
SDTHQOXRWZXTJF
|
6.2 | Ki | 16 | — | |
TVLFEDKEAOXRCZ
|
6.2 | Ki | 22 | — | |
VSVWQTDDGQSGHP
|
6.2 | Ki | 51 | — | |
XTVULKIROSNNTG
|
6.2 | Ki | 29 | — | |
UBPYILGKFZZVDX
|
6.2 | Kd | 130 | Yes | |
KGXBCWANASZZQG
|
6.2 | IC50 | 5 | — | |
WWDLVMCJDNTBPK
|
6.1 | IC50 | 3 | — | |
CPKWRHVMDOSXKE
|
6.1 | IC50 | 5 | — | |
GSRHFOYGPWJXII
|
6.1 | IC50 | 2 | — | |
DKXHSOUZPMHNIZ
|
6.1 | Ki | 51 | Yes | |
GWXPHWSUMLUDPO
|
6.1 | Ki | 11 | — | |
IYOZTVGMEWJPKR
|
6.1 | Ki | 10 | — | |
QVNZKVACBBTKSL
|
6.1 | Ki | 38 | — | |
SYLTYCLPHHSEIJ
|
6.1 | Ki | 27 | — | |
XKFTZKGMDDZMJI
|
6.1 | Ki | 56 | — | |
ZHNDVKCPJRLARD
|
6.1 | Ki | 3 | — | |
ZLHFILGSQDJULK
|
6.1 | Ki | 37 | Yes | |
PIQCTGMSNWUMAF
|
6.1 | Kd | 137 | Yes | |
JOOXLOJCABQBSG
|
6.0 | Kd | 139 | — | |
ODPGGGTTYSGTGO
|
6.0 | Kd | 153 | — | |
RITAVMQDGBJQJZ
|
6.0 | Kd | 43 | — | |
BIIVYFLTOXDAOV
|
6.0 | Ki | 31 | — | |
BIIVYFLTOXDAOV
|
6.0 | Kd | 82 | Yes | |
GKODJBVKKLQMEY
|
6.0 | Ki | 10 | — | |
HZJDBCYRQSJNLZ
|
6.0 | Ki | 7 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
IYOZTVGMEWJPKR
|
6.0 | IC50 | 5 | — | |
JOGKUKXHTYWRGZ
|
6.0 | Ki | 28 | — | |
LBVKEEFIPBQIMD
|
6.0 | Ki | 27 | — | |
LDHYCINFJPCBRY
|
6.0 | Ki | 9 | — | |
LHQWPYOYDRVMFI
|
6.0 | Ki | 21 | — | |
NKEUPUJTVALZIK
|
6.0 | Ki | 28 | — | |
NMHMCXTYPRADBA
|
6.0 | Ki | 20 | — | |
RTYJMUXLFRYRBU
|
6.0 | Ki | 35 | — | |
ZBYGBITZFKOQTA
|
6.0 | Ki | 18 | — |