Target Details
| UniProt AC | Q5S007 |
|---|---|
| Gene Symbol | LRRK2 |
| Protein Name | Leucine-rich repeat serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23745 (ANK_LRRK2) PF23744 (ARM_LRRK2) PF23748 (Beta-prop_LRRK2) PF16095 (COR-A) PF25497 (COR-B) PF13855 (LRR_8) PF00069 (Pkinase) PF08477 (Roc) |
Summary
- Multi-target molecules 299
- Clinical molecules 21
- Avg pChEMBL 7.24
KEGG Pathways (2)
Associated Diseases (3)
Active Molecules (299)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JYCUVOXSZBECAY
|
6.7 | IC50 | 6 | Yes | |
PHXJVRSECIGDHY
|
6.7 | IC50 | 59 | — | |
UJLAWZDWDVHWOW
|
6.7 | Ki | 11 | — | |
VTQQYBGURNVVFE
|
6.7 | Ki | 17 | — | |
LIEUQFMVFKJKHX
|
6.7 | Kd | 10 | — | |
AWDORCFLUJZUQS
|
6.6 | IC50 | 7 | — | |
DVWFMBFZDOBWAD
|
6.6 | Ki | 8 | — | |
IFPPYSWJNWHOLQ
|
6.6 | Ki | 52 | Yes | |
LRZYYIZFBXFSJB
|
6.6 | Ki | 69 | — | |
UAUJVWLUSNTVTA
|
6.6 | IC50 | 6 | — | |
UIRCQOKSJDLYBB
|
6.6 | Ki | 50 | — | |
GUBJNPWVIUFSTR
|
6.6 | Kd | 103 | — | |
BNSPEWBMGVWZFC
|
6.6 | IC50 | 7 | — | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
YYTFTZONXCQXLW
|
6.5 | IC50 | 3 | — | |
YMIKAQYPFQWUEM
|
6.5 | Ki | 7 | — | |
FHIVNWJIENRJBH
|
6.5 | Ki | 9 | — | |
RKUKAACYUCUJEE
|
6.5 | Ki | 58 | — | |
ZCCJKVBTHCOISJ
|
6.5 | Ki | 46 | — | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
ZQUIUVSYHRHZHW
|
6.5 | IC50 | 2 | — | |
OXSKLFUMHBJZNS
|
6.5 | IC50 | 2 | — | |
ASUXILMTDDVWPD
|
6.5 | Ki | 7 | — | |
HZTYDQRUAWIZRE
|
6.5 | Kd | 40 | Yes | |
SEZFNTZQMWJIAI
|
6.5 | Ki | 22 | — | |
WVDQWAPBMCRMGM
|
6.4 | IC50 | 2 | — | |
DPRNXTSMYVCYLJ
|
6.4 | IC50 | 13 | — | |
HXESDBWWDYJEJQ
|
6.4 | Ki | 10 | — | |
JDIZUWGLJSYCHD
|
6.4 | IC50 | 5 | — | |
LZXPYCSHIFEZMR
|
6.4 | Ki | 4 | — | |
QBKUOOQFSVMDPB
|
6.4 | Ki | 31 | — | |
QNLMLEYLZSGBHP
|
6.4 | Ki | 8 | — | |
WAKGEHXTOOFEAE
|
6.4 | Ki | 27 | — | |
NFNBVXVXMQZSGB
|
6.4 | IC50 | 3 | — | |
LOYSOCNFHOPWJA
|
6.4 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
6.3 | Ki | 44 | — | |
KDLLVDABAMKMLD
|
6.3 | Ki | 4 | — | |
MIJMZVTYIXYSDK
|
6.3 | Ki | 4 | — | |
OMZCMEYTWSXEPZ
|
6.3 | Kd | 43 | Yes | |
QCOULMVHIHJKFY
|
6.3 | Ki | 14 | — | |
RRAMBEGOYIJQHY
|
6.3 | Ki | 11 | — | |
RUPJOKGREQMQSI
|
6.3 | Ki | 9 | — | |
ZGZVRPRSFXRGCF
|
6.3 | Ki | 76 | — | |
BCZRYISUUHVFEC
|
6.3 | IC50 | 2 | — | |
CFTUNRCBCCNBLL
|
6.3 | IC50 | 2 | — | |
COWHLOGPEGRMOS
|
6.3 | IC50 | 2 | — | |
JAXPOXBSVKSIEC
|
6.3 | IC50 | 2 | — | |
JWOJVNKGVGVDHF
|
6.3 | IC50 | 2 | — | |
LWFQFYJPBNDMKL
|
6.3 | IC50 | 2 | — | |
MJXOANVGMNJWLC
|
6.3 | IC50 | 2 | — |