Target Details
| UniProt AC | Q5S007 |
|---|---|
| Gene Symbol | LRRK2 |
| Protein Name | Leucine-rich repeat serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23745 (ANK_LRRK2) PF23744 (ARM_LRRK2) PF23748 (Beta-prop_LRRK2) PF16095 (COR-A) PF25497 (COR-B) PF13855 (LRR_8) PF00069 (Pkinase) PF08477 (Roc) |
Summary
- Multi-target molecules 299
- Clinical molecules 21
- Avg pChEMBL 7.24
KEGG Pathways (2)
Associated Diseases (3)
Active Molecules (299)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
REPCEIPSIPNRSG
|
7.2 | IC50 | 3 | — | |
NVINUNQBDNEMSY
|
7.2 | Ki | 4 | — | |
NVRXTLZYXZNATH
|
7.2 | Ki | 47 | Yes | |
VKBFHTIUXUCYRQ
|
7.2 | Ki | 66 | — | |
LGLHCXISMKHLIK
|
7.2 | IC50 | 3 | — | |
XBTMBRMHZRXXHS
|
7.2 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
7.1 | Kd | 151 | — | |
JIRRPWVFUBYRKX
|
7.1 | IC50 | 5 | — | |
KDKUVYLMPJIGKA
|
7.1 | Ki | 91 | Yes | |
URNZTLZSAVLTIZ
|
7.1 | Ki | 26 | — | |
CJXPNZXEEPSZHK
|
7.1 | IC50 | 5 | — | |
HEZSSKBBLQBTMF
|
7.0 | IC50 | 4 | — | |
HFNKQEVNSGCOJV
|
7.0 | Ki | 18 | — | |
KJMURTHIPWRIMC
|
7.0 | IC50 | 7 | — | |
NGSRRJBACKDZHY
|
7.0 | IC50 | 3 | — | |
ATGVCJYHNOSZEV
|
7.0 | Ki | 23 | — | |
DFMCXVONDDGQIY
|
7.0 | Ki | 66 | — | |
DPEXRCOBPACFOO
|
7.0 | Ki | 36 | — | |
LUPCHAFIKZSOOK
|
7.0 | Ki | 15 | — | |
MBZXMVKLFZXZRB
|
7.0 | IC50 | 4 | — | |
MMFBBQQGBVPLQQ
|
7.0 | Ki | 13 | — | |
RGNHKJWHFIPHIM
|
7.0 | Ki | 66 | — | |
XWEWXOXVGICYJP
|
7.0 | IC50 | 2 | — | |
QMQJFRBEIOAQNT
|
6.9 | IC50 | 3 | — | |
TZWUTAYHWCWNFP
|
6.9 | IC50 | 3 | — | |
UOVCGJXDGOGOCZ
|
6.9 | Ki | 59 | — | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
ZGDYBJXDIXVTLV
|
6.9 | Ki | 54 | — | |
LZQQEGBCKOIYIP
|
6.9 | IC50 | 4 | — | |
WVYPOHDPGYBAGO
|
6.9 | IC50 | 4 | — | |
GQERVRMWWVZZDB
|
6.9 | IC50 | 2 | — | |
JVSJTGAAAMSIAW
|
6.8 | IC50 | 2 | — | |
AUDNGNGLLRZLDR
|
6.8 | Ki | 33 | — | |
FFPHMUIGESPOTK
|
6.8 | IC50 | 6 | — | |
HDRLAVNNWSHSOA
|
6.8 | Ki | 19 | — | |
HFNKQEVNSGCOJV
|
6.8 | Kd | 65 | — | |
IJRBJCMLWLFMIN
|
6.8 | Ki | 17 | — | |
MCKPYPWHBUXLEZ
|
6.8 | Ki | 21 | — | |
MZDKLVOWGIOKTN
|
6.8 | Ki | 80 | — | |
NPRYKZQCTXZUKH
|
6.8 | IC50 | 2 | — | |
ZDPGLLQANLROFM
|
6.8 | Ki | 17 | — | |
XLFNLJYGUOLEJS
|
6.8 | IC50 | 26 | — | |
ZQLRNXSQXQGVBK
|
6.8 | Ki | 7 | — | |
XVBGRTMNFNMINE
|
6.8 | IC50 | 5 | — | |
MUMGBSXQGWFWJQ
|
6.8 | IC50 | 2 | — | |
YISURKKUAGVOIV
|
6.8 | IC50 | 2 | — | |
VWYUDOILCXXTFT
|
6.7 | IC50 | 5 | — | |
CNFLHWVYIFARIM
|
6.7 | Ki | 7 | — | |
BLQYVHBZHAISJM
|
6.7 | Ki | 54 | — | |
CRKQBJZCCHKEGI
|
6.7 | Ki | 20 | — |