Target Details
| UniProt AC | Q5S007 |
|---|---|
| Gene Symbol | LRRK2 |
| Protein Name | Leucine-rich repeat serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23745 (ANK_LRRK2) PF23744 (ARM_LRRK2) PF23748 (Beta-prop_LRRK2) PF16095 (COR-A) PF25497 (COR-B) PF13855 (LRR_8) PF00069 (Pkinase) PF08477 (Roc) |
Summary
- Multi-target molecules 299
- Clinical molecules 21
- Avg pChEMBL 7.24
KEGG Pathways (2)
Associated Diseases (3)
Active Molecules (299)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YEVOZZZLKJKCCD
|
7.7 | IC50 | 2 | — | |
AXVWXYOCYXZGCZ
|
7.7 | IC50 | 3 | — | |
IQNTXIMXKCURDC
|
7.7 | IC50 | 3 | — | |
HGHFBVBNHYJNHK
|
7.6 | IC50 | 3 | — | |
JVVFSGBLMWRDED
|
7.6 | IC50 | 2 | — | |
QSDVZPULRUJSBC
|
7.6 | IC50 | 4 | — | |
PELIWNRKLAFPFO
|
7.6 | IC50 | 3 | — | |
OVLGSAZYDZSQMN
|
7.6 | IC50 | 2 | — | |
JNXJKTXDSPWNRP
|
7.6 | Ki | 30 | — | |
VCFDMLBPASGZTP
|
7.6 | Ki | 38 | — | |
VNDWQCSOSCCWIP
|
7.6 | Ki | 39 | Yes | |
WPHKIQPVPYJNAX
|
7.6 | Ki | 81 | — | |
ZWDUUSQSMVRZHV
|
7.6 | IC50 | 3 | — | |
WMICXYLSLOPNDL
|
7.6 | IC50 | 2 | — | |
DDTPGANIPBKTNU
|
7.5 | IC50 | 8 | — | |
YACNMLLIRLXUQZ
|
7.5 | IC50 | 2 | — | |
OQBJXGADOAMRSR
|
7.5 | IC50 | 5 | — | |
WUWXJIFZTHONGM
|
7.5 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
OUJZYQBEFNDJQN
|
7.5 | Ki | 71 | — | |
VRIFJAKXSBXYFZ
|
7.5 | Ki | 8 | — | |
SAOVTENLRUIQAM
|
7.5 | IC50 | 2 | — | |
HVQAATXUCFUOMV
|
7.5 | IC50 | 2 | — | |
UQHKXSZPEUNUDH
|
7.5 | IC50 | 2 | — | |
TZKBVRDEOITLRB
|
7.4 | IC50 | 7 | — | |
FTKWFHKMPQIDLM
|
7.4 | Ki | 5 | — | |
GJOXRIYWDHESDF
|
7.4 | Ki | 27 | — | |
SWVWXQFAJXFRCG
|
7.4 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
7.4 | IC50 | 201 | Yes | |
XZXHXSATPCNXJR
|
7.4 | Kd | 165 | Yes | |
YDRMVAPJCHICGE
|
7.4 | IC50 | 2 | — | |
LVPXBXFMUREXPT
|
7.3 | IC50 | 2 | — | |
WVOMGQLDVCJODR
|
7.3 | IC50 | 3 | — | |
QZZMUIJVVAGHJA
|
7.3 | IC50 | 3 | — | |
YVKIJUOXNIWLHR
|
7.3 | IC50 | 2 | — | |
SGWLRDAOCLITOM
|
7.3 | IC50 | 7 | — | |
JJGSOVIZOMZMCS
|
7.3 | Ki | 35 | — | |
NCXSLSJEOUOJBB
|
7.3 | IC50 | 3 | — | |
ZLLCVOJWNDZXIO
|
7.3 | Ki | 11 | — | |
AILRADAXUVEEIR
|
7.3 | IC50 | 75 | — | |
MTLHRGZTWNKSBV
|
7.3 | Ki | 5 | — | |
UTBRMMZZLJGOHJ
|
7.3 | IC50 | 2 | — | |
WTBSONAFDKCPEQ
|
7.3 | IC50 | 2 | — | |
NLXGPUYLEYEZDV
|
7.3 | IC50 | 2 | — | |
RMHCPURYCHBPLB
|
7.3 | IC50 | 2 | — | |
WEZBTQCZESWSRP
|
7.3 | IC50 | 2 | — | |
DSGOWECLCGJGIL
|
7.2 | IC50 | 2 | — | |
JGVXSQJYBQAPAE
|
7.2 | IC50 | 3 | — | |
YLFKKEGPGBLFKJ
|
7.2 | IC50 | 2 | — | |
NGFGTMFVWSDFPS
|
7.2 | IC50 | 32 | — |