Target Details
| UniProt AC | Q5S007 |
|---|---|
| Gene Symbol | LRRK2 |
| Protein Name | Leucine-rich repeat serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23745 (ANK_LRRK2) PF23744 (ARM_LRRK2) PF23748 (Beta-prop_LRRK2) PF16095 (COR-A) PF25497 (COR-B) PF13855 (LRR_8) PF00069 (Pkinase) PF08477 (Roc) |
Summary
- Multi-target molecules 299
- Clinical molecules 21
- Avg pChEMBL 7.24
KEGG Pathways (2)
Associated Diseases (3)
Active Molecules (299)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FUMCKNCUEAQHCV
|
8.1 | Ki | 103 | — | |
JCFYYOOCRKTOGG
|
8.1 | IC50 | 3 | — | |
SDBOIBYRBWPIEL
|
8.1 | Ki | 31 | — | |
WHVFDYQCAMPLMS
|
8.1 | Ki | 20 | Yes | |
IWMCPJZTADUIFX
|
8.1 | IC50 | 3 | — | |
QRVNXVTYIYXPER
|
8.1 | IC50 | 3 | — | |
AVQNZSIEXOYAGE
|
8.1 | IC50 | 6 | — | |
KHTCIOWVELAJLF
|
8.1 | IC50 | 2 | — | |
YMNHISNDWVXKND
|
8.1 | IC50 | 3 | — | |
DVEKPOFBEAWBKW
|
8.0 | IC50 | 2 | — | |
TVUWQDLBEOZVOU
|
8.0 | Ki | 41 | — | |
IJRGXRBCVBGGOP
|
8.0 | Ki | 2 | — | |
OFUBWOTWQPAEDG
|
8.0 | IC50 | 6 | — | |
QKKIWEILHCXECO
|
8.0 | IC50 | 24 | — | |
SOAIDXSOSFIZBG
|
8.0 | IC50 | 2 | — | |
CRBYIHNRJBMWTM
|
7.9 | IC50 | 2 | — | |
QYYMQRVJYZKVBE
|
7.9 | IC50 | 2 | — | |
JZTOUVBEZONDKA
|
7.9 | Ki | 80 | — | |
BHTWDJBVZQBRKP
|
7.9 | IC50 | 4 | — | |
ONFLVQULIQDDSN
|
7.9 | IC50 | 3 | — | |
UPSNQHGCEYRORJ
|
7.9 | IC50 | 2 | — | |
ACDBIJKZXKGOFW
|
7.8 | IC50 | 2 | — | |
DDJBEYRDSUCNLT
|
7.8 | IC50 | 4 | — | |
MUOUHNBOXJIELS
|
7.8 | IC50 | 3 | — | |
QNABDSWBQJKBHK
|
7.8 | IC50 | 45 | — | |
XCJXNMGPLVXHMC
|
7.8 | IC50 | 4 | — | |
YSFFGUHMDPYPAW
|
7.8 | IC50 | 3 | — | |
MDHMXWJWNZSMEC
|
7.8 | IC50 | 2 | — | |
BGJUMLIDKBULTP
|
7.8 | IC50 | 2 | — | |
HXZURUMJDIMZJI
|
7.8 | IC50 | 3 | — | |
DWHWHOPFYUJPCQ
|
7.8 | IC50 | 2 | — | |
HZPACYSNLOCDLW
|
7.8 | Ki | 48 | — | |
XUFLBSMTYMFOQH
|
7.8 | Ki | 43 | — | |
ZHMXXVNQAFCXKK
|
7.8 | IC50 | 15 | — | |
PFFIEMXZEROLOA
|
7.8 | IC50 | 2 | — | |
ONZFJXAFBPQUIU
|
7.8 | IC50 | 2 | — | |
BOMYQKRMCGRZSK
|
7.8 | IC50 | 2 | — | |
CTQLDDHACGXLAE
|
7.8 | IC50 | 2 | — | |
HKSBXNVKPFTBIG
|
7.8 | IC50 | 3 | — | |
KHCFKCPXXJQHMH
|
7.7 | IC50 | 5 | — | |
OICKVPGRZUWXPB
|
7.7 | IC50 | 3 | — | |
MHPBLCYPFBBOND
|
7.7 | IC50 | 6 | — | |
VNRCXZCFCYFZQN
|
7.7 | IC50 | 2 | — | |
DWTNLZZEPSCAIH
|
7.7 | Ki | 25 | — | |
JMAPTHRNJHOVDP
|
7.7 | IC50 | 3 | — | |
MOXBIRDHNDMBQV
|
7.7 | Ki | 2 | — | |
PRRYQINUAIQTFJ
|
7.7 | Ki | 11 | — | |
QSDVZPULRUJSBC
|
7.7 | IC50 | 3 | — | |
RITAVMQDGBJQJZ
|
7.7 | Ki | 33 | — | |
UYNNRABFCDICBU
|
7.7 | IC50 | 2 | — |