Target Details
| UniProt AC | Q5S007 |
|---|---|
| Gene Symbol | LRRK2 |
| Protein Name | Leucine-rich repeat serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23745 (ANK_LRRK2) PF23744 (ARM_LRRK2) PF23748 (Beta-prop_LRRK2) PF16095 (COR-A) PF25497 (COR-B) PF13855 (LRR_8) PF00069 (Pkinase) PF08477 (Roc) |
Summary
- Multi-target molecules 299
- Clinical molecules 21
- Avg pChEMBL 7.24
KEGG Pathways (2)
Associated Diseases (3)
Active Molecules (299)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IUWWRSQCDUQDEZ
|
12.0 | IC50 | 9 | — | |
OWRXHGAFWZFFCW
|
9.5 | Ki | 113 | — | |
HKSZLNNOFSGOKW
|
9.4 | Ki | 118 | — | |
RYYNGWLOYLRZLK
|
9.2 | Ki | 104 | — | |
ZPPUMAMZIMPJGP
|
9.2 | Ki | 3 | — | |
UJBJWYNPUOLFIZ
|
9.1 | Ki | 49 | — | |
ATUUNJCZCOMUKD
|
9.0 | IC50 | 7 | — | |
HAZVCDSGCISCHC
|
9.0 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
9.0 | IC50 | 49 | Yes | |
PROLIXHVRCJEFH
|
8.9 | Ki | 46 | — | |
VTYLNQMEAHCYTE
|
8.8 | IC50 | 2 | — | |
CLGWUCNXOBLWFM
|
8.8 | IC50 | 2 | — | |
RDHCLVFMADHPEQ
|
8.8 | IC50 | 2 | — | |
HRRUGRNBEPWHFW
|
8.8 | IC50 | 2 | — | |
HRRUGRNBEPWHFW
|
8.8 | IC50 | 2 | — | |
JKIDUHXOZVXHEI
|
8.7 | IC50 | 2 | — | |
PJYWIMRIBDTXII
|
8.7 | IC50 | 2 | — | |
WDARYLSSWBWVCU
|
8.7 | Ki | 49 | — | |
YUKWHAZRUFATPE
|
8.7 | IC50 | 2 | — | |
ONQYZCIVDNVJRE
|
8.6 | Ki | 2 | — | |
ACPZEELFGRNYMY
|
8.6 | IC50 | 2 | — | |
UYJNQQDJUOUFQJ
|
8.6 | Ki | 68 | — | |
QFKKWZVCSJUTOA
|
8.6 | IC50 | 2 | — | |
RKGQENOGQBXEPA
|
8.5 | IC50 | 6 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
ZUOYPKKUCQORTM
|
8.5 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
HKSZLNNOFSGOKW
|
8.4 | IC50 | 408 | — | |
NSGBWKVTGDJMAI
|
8.4 | IC50 | 2 | — | |
BUMVKPFMQPYNEV
|
8.4 | IC50 | 3 | — | |
CPHGZDSYMREPNQ
|
8.4 | IC50 | 6 | — | |
VVPYTOVXFOGRIN
|
8.4 | IC50 | 2 | — | |
JXJKUINEFTUSOV
|
8.4 | IC50 | 2 | — | |
DFBYFJSXUCUKLA
|
8.3 | IC50 | 2 | — | |
GBGQVKUZCXSIOV
|
8.3 | IC50 | 2 | — | |
MFHHFNYSUNIIMQ
|
8.3 | IC50 | 2 | — | |
UWHQAHZPBAISBU
|
8.3 | IC50 | 2 | — | |
XJNDWYLNOREHCQ
|
8.3 | IC50 | 2 | — | |
ISCJKSNXTHTNBW
|
8.2 | IC50 | 4 | — | |
AMQCBROKDRYSQO
|
8.2 | Ki | 2 | — | |
PDQWWZCYXKWWON
|
8.2 | IC50 | 2 | — | |
UYRIPPKFZHHKOO
|
8.2 | Ki | 2 | — | |
WJQKDQRBBJAHPX
|
8.2 | Ki | 2 | — | |
ZPYKCIFIFZRSDS
|
8.2 | Ki | 2 | — | |
KCMYPBPMTXEKNF
|
8.2 | IC50 | 7 | — | |
NWMPVMMGSHXANZ
|
8.2 | Ki | 58 | — | |
CNYOFMNBFMTOHX
|
8.2 | IC50 | 5 | — | |
CRFHZXHUGPCWJA
|
8.2 | IC50 | 8 | — | |
OUDNHJQPMQFCDI
|
8.2 | IC50 | 4 | — | |
QQWUGDVOUVUTOY
|
8.1 | IC50 | 231 | Yes |