Target Details
| UniProt AC | Q5EI73 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Plasmodium falciparum |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 32
- Clinical molecules 8
- Avg pChEMBL 8.17
Active Molecules (32)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SPEKKKWCEBGMGP
|
9.4 | IC50 | 2 | — | |
IDHGAQOVWWBGFK
|
9.3 | IC50 | 4 | — | |
JNJBXYHGNTUTTK
|
9.2 | IC50 | 4 | Yes | |
VLQSBTGRKZOYFJ
|
9.2 | IC50 | 4 | Yes | |
YHWHZGNJXZQUQM
|
9.2 | IC50 | 5 | — | |
UUXJPDYOJAJQGO
|
9.1 | IC50 | 4 | — | |
NLCBWQRVYLSINY
|
9.1 | IC50 | 4 | Yes | |
MBTVJGVVXHCRCZ
|
9.0 | IC50 | 2 | — | |
GGKUJNMJJNAMPQ
|
8.9 | IC50 | 2 | — | |
LNNRPGCPPFJQSP
|
8.8 | IC50 | 4 | — | |
WJNQCZYLIZZQGJ
|
8.7 | IC50 | 2 | — | |
IJCDWDJDJPZXSX
|
8.7 | IC50 | 5 | — | |
MRIVPRZNMCCALI
|
8.7 | IC50 | 2 | — | |
GQLZRVHYGCXHSR
|
8.6 | IC50 | 4 | — | |
UJRBNGYJDIGSOL
|
8.3 | IC50 | 5 | — | |
SAVLZOMOKUOGAK
|
8.3 | IC50 | 2 | — | |
CAZKPPOQQJGGBL
|
8.1 | IC50 | 4 | Yes | |
OLCWFLWEHWLBTO
|
8.1 | IC50 | 2 | — | |
VCBCUVKYTUDCRS
|
8.1 | IC50 | 4 | — | |
OHMYEZKFMQAYKQ
|
8.1 | IC50 | 5 | — | |
ROYSOBXGDVHDTQ
|
8.1 | IC50 | 5 | Yes | |
KULAYTGUTXCHSV
|
7.8 | IC50 | 4 | Yes | |
PLHJCIYEEKOWNM
|
7.8 | IC50 | 4 | Yes | |
RLPQEDLXFSQTGA
|
7.5 | IC50 | 4 | — | |
YQWVLANNJBATDL
|
7.4 | IC50 | 2 | — | |
PLJBZEPECJYWNJ
|
7.3 | IC50 | 4 | — | |
UQPBEYBGEYZEHF
|
7.3 | IC50 | 4 | — | |
VYLMFRUDZGQCNT
|
7.2 | IC50 | 6 | Yes | |
UTULHUYCFSMXCU
|
7.0 | IC50 | 4 | — | |
BFHSSSJPOOPPJC
|
6.8 | IC50 | 4 | — | |
MUGOBVVTADQYDA
|
6.6 | IC50 | 2 | — | |
UIOVGRXEBWMUQT
|
6.0 | IC50 | 2 | — |