Target Details
| UniProt AC | Q59H18 |
|---|---|
| Gene Symbol | TNNI3K |
| Protein Name | Serine/threonine-protein kinase TNNI3K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 122
- Clinical molecules 8
- Avg pChEMBL 7.24
Associated Diseases (1)
Active Molecules (122)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FJUSMFQKFHWCSX
|
6.7 | IC50 | 2 | — | |
GXUZZZRWJPJLHA
|
6.7 | IC50 | 2 | — | |
WTUQKICTFCBUOL
|
6.7 | IC50 | 2 | — | |
RAHBGWKEPAQNFF
|
6.7 | Kd | 26 | — | |
CVKDTMOMVBGJJS
|
6.7 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
6.5 | Kd | 85 | Yes | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
HHZIURLSWUIHRB
|
6.4 | Kd | 57 | Yes | |
PLVDPVQBUNFANZ
|
6.4 | IC50 | 2 | — | |
UQRDFVIQXQYGGX
|
6.4 | IC50 | 2 | — | |
YOTYCNYCVNOPGO
|
6.4 | IC50 | 2 | — | |
ONVDHHGLDDAZRU
|
6.3 | IC50 | 2 | — | |
VGQHMTSLJFXLBO
|
6.3 | IC50 | 2 | — | |
AAKJLRGGTJKAMG
|
6.2 | Kd | 50 | Yes | |
DBGUFUJBJDNCPS
|
6.1 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.1 | Kd | 200 | — | |
MFAQYJIYDMLAIM
|
6.1 | Kd | 130 | Yes | |
HKSZLNNOFSGOKW
|
6.0 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.0 | Kd | 213 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |