Target Details
| UniProt AC | Q59H18 |
|---|---|
| Gene Symbol | TNNI3K |
| Protein Name | Serine/threonine-protein kinase TNNI3K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 122
- Clinical molecules 8
- Avg pChEMBL 7.24
Associated Diseases (1)
Active Molecules (122)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTJOQDUGAGFHMY
|
7.4 | IC50 | 2 | — | |
KERBJUHOPWFOPV
|
7.4 | IC50 | 4 | — | |
QMRCGCBWNRHDTC
|
7.4 | IC50 | 2 | — | |
SIIQKZPELCBJKV
|
7.4 | IC50 | 4 | — | |
UCBHSPGNEZCSHN
|
7.4 | IC50 | 2 | — | |
DXBSLZLNIUZIQJ
|
7.3 | IC50 | 3 | — | |
VAARYSWULJUGST
|
7.3 | Kd | 119 | Yes | |
CGGLCGPBRBEBNW
|
7.3 | IC50 | 2 | — | |
DDDLGNOZDKDSEG
|
7.3 | IC50 | 4 | — | |
FRRDBCZMMUBGNF
|
7.3 | IC50 | 2 | — | |
GUMKQZCYHBFLDF
|
7.3 | IC50 | 4 | — | |
HSXXPAFGNVISQH
|
7.3 | IC50 | 2 | — | |
QMWVXRWLWOVZNH
|
7.3 | IC50 | 4 | — | |
VHHKKIFOCYZSOY
|
7.3 | IC50 | 3 | — | |
YJPQMIQMTGFJMV
|
7.3 | IC50 | 2 | — | |
YZKRTLLFUBQEHG
|
7.3 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
7.3 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
7.3 | Kd | 82 | Yes | |
APTZOLCMZQNBAH
|
7.2 | IC50 | 2 | — | |
BUJLMFKZIJWAPL
|
7.2 | IC50 | 4 | — | |
GIUIYYXTYIIFDX
|
7.2 | IC50 | 4 | — | |
ICLSHNIWDHMQDD
|
7.2 | IC50 | 2 | — | |
NRHLZORMVVHHTO
|
7.2 | IC50 | 2 | — | |
POLFXEZBQNZFED
|
7.2 | IC50 | 2 | — | |
VFTOJSGZOBTVNY
|
7.2 | IC50 | 4 | — | |
WDWFOYNZUZNVNJ
|
7.2 | IC50 | 2 | — | |
AAOSTHUYAHBMNL
|
7.1 | IC50 | 2 | — | |
BAIIHZVEJPNISD
|
7.1 | IC50 | 3 | — | |
FFRWTFPJRTXJRL
|
7.1 | IC50 | 2 | — | |
OOBRVBGRWPCKGK
|
7.1 | IC50 | 2 | — | |
PEIKXUOEORFVSB
|
7.1 | IC50 | 2 | — | |
WFTZMAAMCVPJJT
|
7.1 | IC50 | 26 | — | |
TUINBAPNAKPWHO
|
7.0 | IC50 | 2 | — | |
FLWDQXQPTMVOLP
|
7.0 | IC50 | 2 | — | |
FNRKRAHEJJODJT
|
7.0 | IC50 | 2 | — | |
GRKHWSIIZZRHBT
|
7.0 | IC50 | 2 | — | |
RQNWKCHEEKHWBJ
|
7.0 | IC50 | 2 | — | |
UNTAIBDOCLMZCM
|
7.0 | IC50 | 2 | — | |
ZQKJYEGULARCAH
|
7.0 | IC50 | 3 | — | |
KTEIFNKAUNYNJU
|
7.0 | Kd | 114 | — | |
ARMYNGCDLOKDLO
|
6.9 | IC50 | 2 | — | |
BROIYLJWUMQYQV
|
6.9 | IC50 | 2 | — | |
MGDKKLPMXIEOJN
|
6.9 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
6.9 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.9 | Kd | 149 | — | |
AYUVTOFTSPATMT
|
6.8 | IC50 | 2 | — | |
GKEWVEBUWAKAFT
|
6.8 | IC50 | 3 | — | |
UFOWTGKMZRYQED
|
6.8 | IC50 | 4 | — | |
ODPGGGTTYSGTGO
|
6.8 | Kd | 153 | — | |
UBPYILGKFZZVDX
|
6.8 | Kd | 130 | Yes |