Target Details
| UniProt AC | Q58F21 |
|---|---|
| Gene Symbol | BRDT |
| Protein Name | Bromodomain testis-specific protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 211
- Clinical molecules 0
- Avg pChEMBL 7.28
Associated Diseases (1)
Active Molecules (211)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NETXMUIMUZJUTB
|
6.2 | IC50 | 4 | — | |
IRXGEPQYGSUCML
|
6.1 | IC50 | 3 | — | |
GVJYOLRRZZUUOE
|
6.1 | Kd | 5 | — | |
QUHZSJOJWWZZCP
|
6.1 | IC50 | 4 | — | |
JNPLKPXUKXLWKV
|
6.1 | Ki | 2 | — | |
IQHRPUHKLPCOKF
|
6.1 | Kd | 2 | — | |
QAXOLKUTJAQVHO
|
6.0 | IC50 | 3 | — | |
XWNHXTVCPNRSTM
|
6.0 | IC50 | 3 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |