Target Details
| UniProt AC | Q58F21 |
|---|---|
| Gene Symbol | BRDT |
| Protein Name | Bromodomain testis-specific protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 211
- Clinical molecules 0
- Avg pChEMBL 7.28
Associated Diseases (1)
Active Molecules (211)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UCJMBWXOKLINTN
|
6.7 | Kd | 4 | — | |
FRBRZGLUFOZRGD
|
6.7 | IC50 | 4 | — | |
NGXAMXNWIHBLBN
|
6.7 | Kd | 6 | — | |
JCGSQIXZALUTFO
|
6.7 | IC50 | 2 | — | |
ZGOPGBNZFMGVAJ
|
6.7 | IC50 | 2 | — | |
CBJPXYZHTAENCD
|
6.7 | IC50 | 2 | — | |
OABQDWQBXSGEDG
|
6.7 | IC50 | 9 | — | |
GKMMNQCWGZRQTN
|
6.7 | IC50 | 4 | — | |
JVAKWUYUZCOCKR
|
6.7 | IC50 | 4 | — | |
RSMYFSPOTCDHHJ
|
6.7 | Ki | 5 | — | |
DYQPKOGFUIEBMS
|
6.6 | IC50 | 3 | — | |
HFXQHVKVUNQRBN
|
6.6 | IC50 | 7 | — | |
KXSJLOFFUFDGTE
|
6.6 | IC50 | 6 | — | |
OBZUUWUBOOUBNE
|
6.6 | IC50 | 7 | — | |
DGJREYHVQYZTEV
|
6.6 | Kd | 6 | — | |
HTPNGOWITIWAHM
|
6.6 | IC50 | 3 | — | |
XQVVPGYIWAGRNI
|
6.6 | Kd | 34 | — | |
IHOWNNYVAUSWOU
|
6.6 | IC50 | 7 | — | |
MTBDHPJCWYLCBM
|
6.5 | IC50 | 7 | — | |
LBXYVUXGPFEVSI
|
6.5 | IC50 | 3 | — | |
ZGCHTGGUXZBHCN
|
6.5 | IC50 | 7 | — | |
JOOXLOJCABQBSG
|
6.5 | IC50 | 139 | — | |
IZLQRTZZHBLSKO
|
6.5 | IC50 | 6 | — | |
DYQPKOGFUIEBMS
|
6.5 | IC50 | 3 | — | |
FSMTUHGXWGJNKK
|
6.5 | IC50 | 4 | — | |
XOCKWBJNBUYYAL
|
6.5 | IC50 | 5 | — | |
ZBRDRGVJFCJFQS
|
6.5 | IC50 | 2 | — | |
CFTIJALKSHXVNU
|
6.4 | IC50 | 3 | — | |
IRCDNPBWELYZBD
|
6.4 | IC50 | 3 | — | |
DJNZZLZKAXGMMC
|
6.4 | Kd | 3 | — | |
VBDIOKSSYUZONA
|
6.4 | IC50 | 3 | — | |
VLSYQVCLFAZVNI
|
6.4 | IC50 | 2 | — | |
BHUOTMULUBCHII
|
6.4 | IC50 | 3 | — | |
MWNUDTXWOMXGKW
|
6.3 | IC50 | 2 | — | |
IPZXGSLENCVPEZ
|
6.3 | IC50 | 2 | — | |
DQFBZYXAVHHSEQ
|
6.3 | IC50 | 2 | — | |
JGGBFOUTSJEGRT
|
6.3 | Ki | 4 | — | |
XVBGRTMNFNMINE
|
6.3 | Kd | 5 | — | |
GHYCWVRIEDGGFQ
|
6.3 | IC50 | 4 | — | |
GVCFSBGCJBRHFS
|
6.3 | IC50 | 4 | — | |
IWMCPJZTADUIFX
|
6.3 | Kd | 3 | — | |
BROHMTOMOQOASI
|
6.2 | IC50 | 2 | — | |
ITDUQSWFIDASGI
|
6.2 | IC50 | 3 | — | |
YGQSAYAQCWLSAL
|
6.2 | IC50 | 3 | — | |
VYSDIFXQJTUSHB
|
6.2 | IC50 | 2 | — | |
DIVYGZNYLRPCMD
|
6.2 | IC50 | 2 | — | |
IUCHPMDFWMIAJM
|
6.2 | IC50 | 2 | — | |
NIFODZUHQBXOII
|
6.2 | IC50 | 6 | — | |
MVMMNLALSKWQDY
|
6.2 | IC50 | 2 | — | |
MUOCQMZJLRQTRD
|
6.2 | Ki | 2 | — |