Target Details
| UniProt AC | Q58F21 |
|---|---|
| Gene Symbol | BRDT |
| Protein Name | Bromodomain testis-specific protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 211
- Clinical molecules 0
- Avg pChEMBL 7.28
Associated Diseases (1)
Active Molecules (211)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZXGRKOXAZLNTEL
|
7.2 | IC50 | 2 | — | |
ARWMKZDWGIOCEU
|
7.2 | IC50 | 4 | — | |
AULNYQHQUIEHMG
|
7.2 | IC50 | 2 | — | |
POKZINYHLOHGEB
|
7.2 | Kd | 4 | — | |
QTVSDAUHDJBCAA
|
7.2 | IC50 | 4 | — | |
JQGLKQWMMRCIIG
|
7.2 | IC50 | 4 | — | |
SKANTSCEPLCAJH
|
7.2 | IC50 | 2 | — | |
SKANTSCEPLCAJH
|
7.2 | IC50 | 2 | — | |
NHMJYXDPZTZGQX
|
7.1 | IC50 | 2 | — | |
NHMJYXDPZTZGQX
|
7.1 | IC50 | 2 | — | |
DNVXATUJJDPFDM
|
7.1 | IC50 | 4 | — | |
QIEVBHRUPLMWFP
|
7.1 | Kd | 2 | — | |
LEXSRVMWXAFLMV
|
7.1 | IC50 | 4 | — | |
LEXSRVMWXAFLMV
|
7.1 | IC50 | 3 | — | |
XXZLLCKEAYMUHY
|
7.1 | IC50 | 2 | — | |
ZXGRKOXAZLNTEL
|
7.1 | IC50 | 2 | — | |
ZXGRKOXAZLNTEL
|
7.1 | IC50 | 2 | — | |
AAAQFGUYHFJNHI
|
7.1 | Kd | 252 | — | |
FRBRZGLUFOZRGD
|
7.1 | IC50 | 5 | — | |
XQODQNSFZKRZIC
|
7.1 | Kd | 4 | — | |
CYUUSRGILFWDHA
|
7.0 | IC50 | 2 | — | |
QXWJFGXUZLPVCL
|
7.0 | IC50 | 2 | — | |
ZYJNOYAZLFPWBD
|
7.0 | IC50 | 4 | — | |
HIZNONHBBUUYFX
|
7.0 | IC50 | 4 | — | |
DNVXATUJJDPFDM
|
7.0 | IC50 | 2 | — | |
HTPNGOWITIWAHM
|
7.0 | IC50 | 3 | — | |
WWFAGXVFIAJTJE
|
7.0 | IC50 | 2 | — | |
GZFJPALDEYOFHA
|
7.0 | Ki | 6 | — | |
SXNJFOWDRLKDSF
|
7.0 | Kd | 8 | — | |
RQCMHFWZGCIXKC
|
6.9 | IC50 | 2 | — | |
CPTTUKGIGKOQKE
|
6.9 | IC50 | 2 | — | |
SOYMCIQWSHFMKE
|
6.9 | IC50 | 2 | — | |
RXAFLNFTNQFCIB
|
6.9 | IC50 | 2 | — | |
VUVUVNZRUGEAHB
|
6.9 | IC50 | 5 | — | |
CAKYNETUOQZPMX
|
6.9 | IC50 | 2 | — | |
IKKUVCXGUJTONF
|
6.9 | IC50 | 6 | — | |
KXQSVQUUJQXHIX
|
6.9 | IC50 | 2 | — | |
DNVXATUJJDPFDM
|
6.9 | IC50 | 4 | — | |
PKFVMDLBSYTDCI
|
6.8 | IC50 | 2 | — | |
QNOJAPBYTXGBLX
|
6.8 | Ki | 5 | — | |
RXVUXTUHNJFNBM
|
6.8 | IC50 | 2 | — | |
ZLSFDTLLWMDEFA
|
6.8 | IC50 | 2 | — | |
ZORLJXWXFABTPZ
|
6.8 | IC50 | 9 | — | |
SUFVOUWYHJXPBW
|
6.8 | Kd | 4 | — | |
DNVXATUJJDPFDM
|
6.7 | IC50 | 17 | — | |
QZZCUOVXHPAQRQ
|
6.7 | IC50 | 5 | — | |
CAKYNETUOQZPMX
|
6.7 | IC50 | 2 | — | |
GFDDTDKCZCGJLM
|
6.7 | Kd | 5 | — | |
SDIHFORMFMHWNK
|
6.7 | IC50 | 6 | — | |
AJFFVWPPDGTGNY
|
6.7 | IC50 | 2 | — |