Target Details
| UniProt AC | Q58F21 |
|---|---|
| Gene Symbol | BRDT |
| Protein Name | Bromodomain testis-specific protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 211
- Clinical molecules 0
- Avg pChEMBL 7.28
Associated Diseases (1)
Active Molecules (211)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VEPYYWIOIMZOLX
|
7.8 | IC50 | 4 | — | |
XBGAIUVLEXZQMO
|
7.8 | IC50 | 4 | — | |
DMSRRTGRIHHJKS
|
7.7 | IC50 | 4 | — | |
MFKPAAFGGBINQO
|
7.7 | IC50 | 4 | — | |
UIWJGKYIPQKBHV
|
7.7 | IC50 | 4 | — | |
UIWJGKYIPQKBHV
|
7.7 | IC50 | 4 | — | |
YYKYSROKVREYAZ
|
7.7 | IC50 | 4 | — | |
VYNYPLNNLNISCK
|
7.7 | IC50 | 4 | — | |
NDEORODKVUYMFQ
|
7.7 | Kd | 9 | — | |
WSHVXKCBHNIVJO
|
7.7 | IC50 | 4 | — | |
PVOCQBDIXSGBCZ
|
7.7 | IC50 | 2 | — | |
HSAHLMIFPRYVEH
|
7.7 | IC50 | 4 | — | |
XBGAIUVLEXZQMO
|
7.7 | IC50 | 4 | — | |
FXBLOXPPYWAJKD
|
7.7 | IC50 | 2 | — | |
RBZRCEPYYVFROZ
|
7.7 | Kd | 5 | — | |
UXFXOEGGFKVCDW
|
7.6 | IC50 | 4 | — | |
XQSIYYHBLOKYON
|
7.6 | IC50 | 2 | — | |
BRAMSTZRKUJRKS
|
7.6 | IC50 | 4 | — | |
BRAMSTZRKUJRKS
|
7.6 | IC50 | 3 | — | |
KNBYFXZNSOENGW
|
7.6 | Kd | 5 | — | |
OEDSFMUSNZDJFD
|
7.5 | Ki | 4 | — | |
BHEROPFARKLXOP
|
7.5 | IC50 | 4 | — | |
BRBCSVDUUHHTIS
|
7.5 | IC50 | 4 | — | |
PQSJCTLBPAPREX
|
7.5 | IC50 | 2 | — | |
URJBVMXNPKFWPB
|
7.5 | IC50 | 2 | — | |
OTOVUBXMOLCWFF
|
7.5 | IC50 | 2 | — | |
LORVKFYVSXATKW
|
7.5 | IC50 | 5 | — | |
NECWWYRRULAEDN
|
7.5 | IC50 | 2 | — | |
FZFLGRAVZYFGBB
|
7.4 | Kd | 4 | — | |
QSRRNUBIKNVQHO
|
7.4 | Kd | 4 | — | |
PDCBJZVPIGAEBL
|
7.4 | IC50 | 4 | — | |
SADKUQHRGVTPSQ
|
7.4 | IC50 | 4 | — | |
UYBRROMMFMPJAN
|
7.4 | Kd | 8 | — | |
XTJGRKJBJUZZJT
|
7.4 | IC50 | 2 | — | |
MYTABVRHXGACGI
|
7.4 | IC50 | 4 | — | |
NAPOLFVZKFHOBG
|
7.4 | IC50 | 4 | — | |
KTPZIQXMURKYQT
|
7.3 | IC50 | 2 | — | |
LLRPIXCDTAUFLE
|
7.3 | IC50 | 4 | — | |
USNVRJYSAUJTNT
|
7.3 | IC50 | 4 | — | |
JKLFTZFZNNCDAE
|
7.3 | IC50 | 4 | — | |
FAWSUKOIROHXAP
|
7.3 | IC50 | 5 | — | |
MMMRGZLSUKMQOD
|
7.3 | IC50 | 4 | — | |
NHQWTZLQTWSZGU
|
7.3 | IC50 | 4 | — | |
ABSZIZKRSYKAPX
|
7.2 | IC50 | 4 | — | |
SVWVGWHDUPYUFQ
|
7.2 | IC50 | 4 | — | |
JXLHJBYUGDELIZ
|
7.2 | IC50 | 2 | — | |
XLAWIKASUIIZGC
|
7.2 | IC50 | 2 | — | |
GZEDEKFDZMUCGJ
|
7.2 | IC50 | 4 | — | |
PIKWYDHWUKSWAQ
|
7.2 | Kd | 4 | — | |
ZXGRKOXAZLNTEL
|
7.2 | IC50 | 2 | — |