Target Details
UniProt ACQ58F21
Gene SymbolBRDT
Protein NameBromodomain testis-specific protein
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain)
Summary
  • Multi-target molecules 211
  • Clinical molecules 0
  • Avg pChEMBL 7.28
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (211)
InChIKey pChEMBL Type Targets Clinical
JNSLBXJNVHYNNW 10.1 Ki 4
VGOFJMULWAVDMV 10.1 Kd 2
LMLIBNUOIWAJFC 9.6 Kd 9
FZWPGKYEENZFAU 9.5 Ki 4
LJLJARSDBHJRGG 9.2 Ki 4
VLYMRIROHVATMC 9.1 Kd 2
YTJRGAPMTDBXIK 9.1 Kd 2
YQUPOPCILRFMSA 9.1 IC50 2
KYCQRWFJRCYKBU 9.0 IC50 2
DPQKUYBPPCXREN 8.9 Kd 2
AMHWRJBEKUEFFO 8.8 Kd 2
WHJGVHRMVTVKHR 8.8 IC50 2
OPVRCPHGQNNHNN 8.7 IC50 2
JIYPVUCBRQNICX 8.7 Kd 7
KTPZIQXMURKYQT 8.7 IC50 2
UETQFSCWDMJWMM 8.7 Kd 4
RDONXGFGWSSFMY 8.7 Ki 6
NOYKJWSXDSTVCB 8.6 IC50 2
QKJZSKDMERAPEK 8.6 Kd 2
OZPNRBXVIUPSDJ 8.5 Kd 4
FNHHVPPSBFQMEL 8.4 IC50 4
UNODBAFOZVBZBF 8.4 Ki 4
WOHZTCPWKXURKU 8.3 IC50 2
KHQQNXFBTALTQF 8.3 Kd 6
WZQLVEPIBAOOGF 8.3 Kd 9
HKDZBPLAJAVDDD 8.3 IC50 2
UDJIOTIVUUWIDN 8.3 IC50 2
LQNCVLFKDSYCTE 8.2 IC50 2
LKEGXJXRNBALBV 8.2 Kd 5
LMYMWXJBPLXESU 8.2 Kd 2
GHHBKDUDXQGYHF 8.2 IC50 2
ZJKGEINLDGYOLW 8.2 IC50 2
OJSKWCXPUVTNCF 8.2 IC50 4
QMIQDDJVGIKUJA 8.2 IC50 2
KPWWFNXRLAAREN 8.1 Kd 12
AEANZCXROGPSBY 8.0 Kd 6
PHSKNIAWTPPDAY 8.0 IC50 2
RDWRDUFEWMSPGQ 8.0 Kd 4
JBPWXWQIGDWQHR 8.0 IC50 15
WOHDSOWPKUZJTL 7.9 IC50 2
GCDAPUPAGHUHLH 7.9 IC50 4
WOSYEWDDCNUUHT 7.9 IC50 4
AIEAYHRNULRMLO 7.9 IC50 2
GTOKRJQCMDFUOW 7.9 IC50 2
MDRXOFSNECSECW 7.9 Kd 4
RKPWYUDCZHEUBU 7.8 IC50 4
TUDWFCNTNUMOKQ 7.8 IC50 2
GCDAPUPAGHUHLH 7.8 IC50 4
PWEXGFMQMFFMNN 7.8 IC50 4
RJJDAOYTHRXSGL 7.8 IC50 4
2D structure