Target Details
| UniProt AC | Q582G3 |
|---|---|
| Gene Symbol | Tb07.10C21.550 |
| Protein Name | Bifunctional dihydrofolate reductase-thymidylate synthase |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) PF00303 (Thymidylat_synt) |
Summary
- Multi-target molecules 10
- Clinical molecules 1
- Avg pChEMBL 6.48
Top Co-occurrence Targets
- Tb08.26N11.790 10 shared
- 8 shared
- PTR1 7 shared
- DHFR 2 shared
- 1 shared
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBOZXECLQNJBKD
|
8.0 | IC50 | 4 | Yes | |
HEPDQIIFCBFHRJ
|
6.6 | IC50 | 4 | — | |
UKCFUFHREWUXJJ
|
6.6 | IC50 | 5 | — | |
ASBJYAZYFSRQAB
|
6.5 | IC50 | 4 | — | |
NKRKEQBTIYLTPA
|
6.4 | IC50 | 4 | — | |
QVHFSGMRVQZGMC
|
6.3 | IC50 | 4 | — | |
NQLDZGLJAMJTPQ
|
6.2 | IC50 | 3 | — | |
OTZWZUHDCONCKN
|
6.2 | IC50 | 3 | — | |
URXOGQMRRPHSHR
|
6.0 | IC50 | 4 | — | |
CZUHYAFUFAOCJF
|
6.0 | IC50 | 3 | — |