Target Details
| UniProt AC | Q581W1 |
|---|---|
| Gene Symbol | Tb08.26N11.790 |
| Protein Name | N/A |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13561 (adh_short_C2) |
Summary
- Multi-target molecules 30
- Clinical molecules 1
- Avg pChEMBL 7.55
Top Co-occurrence Targets
- PTR1 23 shared
- 13 shared
- Tb07.10C21.550 10 shared
- PTR1 4 shared
- DHFR 2 shared
- 1 shared
Active Molecules (30)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ASBJYAZYFSRQAB
|
10.0 | IC50 | 4 | — | |
FGQMPGXSJKTERW
|
10.0 | IC50 | 3 | — | |
URXOGQMRRPHSHR
|
10.0 | IC50 | 4 | — | |
CZUHYAFUFAOCJF
|
9.0 | IC50 | 3 | — | |
HEPDQIIFCBFHRJ
|
9.0 | IC50 | 4 | — | |
WSVXHZUMXANBHW
|
9.0 | IC50 | 2 | — | |
JFVMZMBFRZPOFF
|
8.2 | Ki | 2 | — | |
LMNKJAVCUDBBQL
|
8.0 | IC50 | 2 | — | |
QVHFSGMRVQZGMC
|
8.0 | IC50 | 4 | — | |
XJIGBPBDYCDOJG
|
8.0 | IC50 | 2 | — | |
AMDVLSYFJVONRJ
|
7.5 | IC50 | 3 | — | |
NKRKEQBTIYLTPA
|
7.5 | IC50 | 4 | — | |
FMBRAYUCAAUXJJ
|
7.4 | IC50 | 3 | — | |
UHGIVIFLYVOBQX
|
7.4 | IC50 | 3 | — | |
ODCTYJXVCFVIBH
|
7.3 | Ki | 2 | — | |
FBOZXECLQNJBKD
|
7.3 | IC50 | 4 | Yes | |
UKCFUFHREWUXJJ
|
7.3 | IC50 | 5 | — | |
OTZWZUHDCONCKN
|
7.0 | IC50 | 3 | — | |
NYNAFINLHQEHKU
|
7.0 | IC50 | 3 | — | |
NQLDZGLJAMJTPQ
|
6.8 | IC50 | 3 | — | |
SWCIFVXOLXOGHA
|
6.8 | IC50 | 2 | — | |
OETPLDVKGKXAKN
|
6.7 | IC50 | 2 | — | |
JFXCDKAYLSVCHK
|
6.7 | IC50 | 2 | — | |
OBAQLSSSQKPYLE
|
6.6 | IC50 | 2 | — | |
CIIGLUKLZVOCMA
|
6.5 | IC50 | 2 | — | |
JBNABAJVIVYIDA
|
6.4 | Ki | 2 | — | |
JGIMDXAWKSVXJR
|
6.3 | Ki | 2 | — | |
BGMTVROBCGUEED
|
6.3 | IC50 | 2 | — | |
KIZAIPYPBOOMIP
|
6.3 | IC50 | 2 | — | |
LMKXBYYGJWCTTQ
|
6.1 | IC50 | 2 | — |