Target Details
| UniProt AC | Q56UN5 |
|---|---|
| Gene Symbol | MAP3K19 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 19 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 59
- Clinical molecules 23
- Avg pChEMBL 7.1
Active Molecules (59)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
9.3 | Kd | 289 | Yes | |
NLGZSRKKPYFWHZ
|
8.9 | Kd | 6 | — | |
HKSZLNNOFSGOKW
|
8.7 | IC50 | 408 | — | |
MFAQYJIYDMLAIM
|
8.3 | Kd | 130 | Yes | |
XZXHXSATPCNXJR
|
8.3 | Kd | 165 | Yes | |
YYLKKYCXAOBSRM
|
8.3 | Kd | 191 | — | |
CXQHYVUVSFXTMY
|
8.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
8.3 | Kd | 149 | — | |
HZRJHVDNTDBTOZ
|
8.0 | Kd | 8 | — | |
CTNPALGJUAXMMC
|
7.9 | Kd | 151 | — | |
PIQCTGMSNWUMAF
|
7.9 | Kd | 137 | Yes | |
BMGQWWVMWDBQGC
|
7.8 | Kd | 147 | Yes | |
JWNPDZNEKVCWMY
|
7.8 | Kd | 57 | Yes | |
UBPYILGKFZZVDX
|
7.8 | Kd | 130 | Yes | |
WINHZLLDWRZWRT
|
7.8 | Kd | 201 | Yes | |
JOOXLOJCABQBSG
|
7.7 | Kd | 139 | — | |
AAKJLRGGTJKAMG
|
7.6 | Kd | 50 | Yes | |
KGPGFQWBCSZGEL
|
7.5 | Kd | 59 | Yes | |
GUBJNPWVIUFSTR
|
7.4 | Kd | 103 | — | |
ZCBUQCWBWNUWSU
|
7.3 | Kd | 59 | — | |
GCIKSSRWRFVXBI
|
7.3 | Kd | 109 | Yes | |
YABJJWZLRMPFSI
|
7.3 | Kd | 34 | — | |
WQVPGYMGERDXLH
|
7.2 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
OYONTEXKYJZFHA
|
7.1 | Kd | 69 | Yes | |
ZBNZXTGUTAYRHI
|
7.1 | Kd | 102 | Yes | |
NENJFZKQHYXRDQ
|
7.0 | Kd | 8 | — | |
BGVLELSCIHASRV
|
7.0 | Kd | 11 | — | |
MLDQJTXFUGDVEO
|
7.0 | Kd | 85 | Yes | |
ODPGGGTTYSGTGO
|
6.9 | Kd | 153 | — | |
BMWMKGNVAMXXCH
|
6.9 | Kd | 6 | — | |
ZZSBPGIGIUFJRA
|
6.9 | Kd | 46 | — | |
ODLDMAFDYHTWSE
|
6.8 | Kd | 5 | — | |
HZTYDQRUAWIZRE
|
6.7 | Kd | 40 | Yes | |
PMDAVRLCSZSLRH
|
6.7 | Kd | 13 | — | |
RAHBGWKEPAQNFF
|
6.7 | Kd | 26 | — | |
JZRNXAPRPJTGOG
|
6.7 | Kd | 3 | — | |
BPNUQXPIQBZCMR
|
6.6 | Kd | 83 | Yes | |
VAARYSWULJUGST
|
6.6 | Kd | 119 | Yes | |
XGALLCVXEZPNRQ
|
6.6 | Kd | 39 | Yes | |
MPVGZUGXCQEXTM
|
6.6 | Kd | 61 | Yes | |
XXJWYDDUDKYVKI
|
6.6 | Kd | 52 | — | |
PSPFQEBFYXJZEV
|
6.6 | Kd | 10 | — | |
HFNKQEVNSGCOJV
|
6.6 | Kd | 65 | — | |
RITAVMQDGBJQJZ
|
6.6 | Kd | 43 | — | |
BGVLELSCIHASRV
|
6.5 | Kd | 12 | — | |
BGVLELSCIHASRV
|
6.5 | Kd | 12 | — | |
FCYPWSQPDXUBPV
|
6.5 | Kd | 2 | — | |
CVWXJKQAOSCOAB
|
6.3 | Kd | 35 | — | |
XQVVPGYIWAGRNI
|
6.3 | Kd | 34 | — |