Target Details
| UniProt AC | Q53GL7 |
|---|---|
| Gene Symbol | PARP10 |
| Protein Name | Protein mono-ADP-ribosyltransferase PARP10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) PF23085 (RRM_PARP14_3) |
Summary
- Multi-target molecules 17
- Clinical molecules 0
- Avg pChEMBL 6.78
Active Molecules (17)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
STSCRAGBCYODMY
|
8.0 | IC50 | 8 | — | |
FSNNMBVVDWKKCB
|
7.5 | IC50 | 6 | — | |
ZKXNKMALIYTLJE
|
7.2 | IC50 | 4 | — | |
KIMPACVVSQUMHL
|
6.9 | IC50 | 2 | — | |
PCAWJIMDNGAMRA
|
6.9 | IC50 | 2 | — | |
JLVRTMBMCWYGAL
|
6.8 | IC50 | 7 | — | |
GJJIICZAOJXOEJ
|
6.8 | IC50 | 2 | — | |
RMIJZTKTCJJVSA
|
6.8 | IC50 | 4 | — | |
MWPKIJXVHHDLCZ
|
6.8 | IC50 | 2 | — | |
RFKWWUGSOVDNFF
|
6.8 | IC50 | 2 | — | |
VQAMGVVQVZCTNJ
|
6.5 | IC50 | 3 | — | |
BMPSOKZAIFFMLK
|
6.5 | IC50 | 6 | — | |
XZRCQWLPMXFGHE
|
6.5 | IC50 | 2 | — | |
FDLYAMZZIXQODN
|
6.4 | IC50 | 11 | — | |
ZXYKQNYSXHNQMV
|
6.4 | IC50 | 6 | — | |
HMABYWSNWIZPAG
|
6.2 | IC50 | 12 | — | |
HTTRFYNWHOXUPE
|
6.1 | IC50 | 3 | — |