Target Details
| UniProt AC | Q4Q5S8 |
|---|---|
| Gene Symbol | NMT |
| Protein Name | Glycylpeptide N-tetradecanoyltransferase |
| Organism | Leishmania major |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01233 (NMT) PF02799 (NMT_C) |
Summary
- Multi-target molecules 90
- Clinical molecules 0
- Avg pChEMBL 7.44
Active Molecules (90)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HLJCVRXGZMOFDS
|
9.2 | IC50 | 4 | — | |
IACHGHVEEMFILS
|
9.0 | IC50 | 3 | — | |
JEXUGPIZWWTQHG
|
9.0 | IC50 | 3 | — | |
PGRFAUBJFXTXLR
|
9.0 | IC50 | 3 | — | |
PPTHDMWUXYOQCC
|
9.0 | IC50 | 3 | — | |
UGQSROIUKTXJQO
|
9.0 | IC50 | 3 | — | |
IMQPHOQRHBIWQQ
|
8.7 | Ki | 2 | — | |
KGUSVAQCTAVWAD
|
8.7 | IC50 | 3 | — | |
LFUKSJMPHXRAHE
|
8.7 | IC50 | 3 | — | |
YMLFRSAHQNBEFS
|
8.6 | Ki | 3 | — | |
NCFHKHWPNGZJEO
|
8.5 | IC50 | 3 | — | |
GLLAAKIAMHKWQW
|
8.4 | IC50 | 3 | — | |
JPEQRKSUSLNASS
|
8.4 | IC50 | 3 | — | |
HAUGBCQQUOZSGH
|
8.3 | IC50 | 3 | — | |
JHFMAYRHBZNEBV
|
8.3 | IC50 | 3 | — | |
PINSRGHFBUSSTB
|
8.3 | IC50 | 3 | — | |
RPZBHCIXTUDXGC
|
8.3 | IC50 | 3 | — | |
RYJPWHHWIOKQFO
|
8.3 | IC50 | 3 | — | |
XANRCBWVKKVBOO
|
8.3 | IC50 | 3 | — | |
XISLEJQCQIHTJT
|
8.3 | IC50 | 3 | — | |
GQRWEJRYCBEXLY
|
8.2 | Ki | 3 | — | |
ADYMPTOMRJWSQN
|
8.1 | Ki | 2 | — | |
KFZNUMAAQRKTIR
|
8.1 | IC50 | 3 | — | |
XMBSZPZJLPTFMV
|
8.0 | Ki | 4 | — | |
DVTQRRNJAIULRN
|
8.0 | IC50 | 3 | — | |
FSQFLTMLOZTAHB
|
8.0 | IC50 | 3 | — | |
GVYHLYWBDITGOO
|
8.0 | IC50 | 3 | — | |
POTVFFXGRINLJD
|
8.0 | IC50 | 3 | — | |
XJHUAHFZFJZMEE
|
7.9 | IC50 | 3 | — | |
KKALBIRLEONXKX
|
7.7 | IC50 | 3 | — | |
PZIZCUMFALUOSC
|
7.7 | IC50 | 3 | — | |
PCURNESJVHMDOH
|
7.7 | Ki | 2 | — | |
GWKJWTPHSUXVCQ
|
7.6 | IC50 | 3 | — | |
AYWNZLSZEHOECC
|
7.6 | Ki | 2 | — | |
COJPRJCSLJKNNT
|
7.6 | IC50 | 3 | — | |
XEIMOGDDPRSYCR
|
7.6 | IC50 | 3 | — | |
RSFRJVKGQDTUAK
|
7.6 | IC50 | 3 | — | |
FGUZNVABRLKYEA
|
7.5 | IC50 | 3 | — | |
GASUPAQGJGLLGM
|
7.5 | IC50 | 3 | — | |
PUVYTKKSEYNATO
|
7.5 | IC50 | 3 | — | |
MZECZFBGNUSGHF
|
7.4 | IC50 | 3 | — | |
OTKMKBYGZQEUCC
|
7.4 | IC50 | 2 | — | |
FHLDEMLNIBTAGL
|
7.4 | IC50 | 3 | — | |
GZQJPTFJBDYKRV
|
7.4 | IC50 | 2 | — | |
IFDWZFPOQYAVFV
|
7.3 | IC50 | 3 | — | |
IXHQESXLKWPGHT
|
7.3 | IC50 | 3 | — | |
OYNUBGTVBHOARA
|
7.3 | IC50 | 3 | — | |
PFWXHLNTKMHYOA
|
7.3 | IC50 | 3 | — | |
XHOICLITTSTOPW
|
7.3 | IC50 | 2 | — | |
YJEDXBAVBHENKZ
|
7.3 | IC50 | 3 | — |