Target Details
| UniProt AC | Q460N5 |
|---|---|
| Gene Symbol | PARP14 |
| Protein Name | Protein mono-ADP-ribosyltransferase PARP14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23084 (KH_PARP14_1) PF23248 (KH_PARP14_2) PF23249 (KH_PARP14_3) PF23251 (KH_PARP14_4) PF23252 (KH_PARP14_5) PF23253 (KH_PARP14_6) PF23254 (KH_PARP14_8) PF01661 (Macro) PF00644 (PARP) PF23222 (RRM_PARP14_1) PF23245 (RRM_PARP14_2) PF23085 (RRM_PARP14_3) PF22005 (WWE_1) |
Summary
- Multi-target molecules 10
- Clinical molecules 0
- Avg pChEMBL 6.32
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GGQAXNFSEUSJJE
|
6.8 | IC50 | 3 | — | |
HIDGSHNRMYFZHS
|
6.6 | IC50 | 2 | — | |
FSNNMBVVDWKKCB
|
6.5 | IC50 | 6 | — | |
DKPIHFWBNZVINS
|
6.4 | IC50 | 2 | — | |
IYJYZOJIOGICFK
|
6.3 | IC50 | 2 | — | |
ZKXNKMALIYTLJE
|
6.2 | IC50 | 4 | — | |
DUVLGZHVLHPLOD
|
6.2 | IC50 | 2 | — | |
UOHKZMQXEJGUES
|
6.2 | IC50 | 4 | — | |
IJTBFOMRKCFLIG
|
6.0 | IC50 | 2 | — | |
RMIJZTKTCJJVSA
|
6.0 | IC50 | 4 | — |