Target Details
| UniProt AC | Q460N3 |
|---|---|
| Gene Symbol | PARP15 |
| Protein Name | Protein mono-ADP-ribosyltransferase PARP15 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01661 (Macro) PF00644 (PARP) |
Summary
- Multi-target molecules 13
- Clinical molecules 0
- Avg pChEMBL 6.49
Active Molecules (13)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FSNNMBVVDWKKCB
|
7.1 | IC50 | 6 | — | |
LQJVOLSLAFIXSV
|
6.6 | IC50 | 4 | — | |
ZKXNKMALIYTLJE
|
6.6 | IC50 | 4 | — | |
VQAMGVVQVZCTNJ
|
6.5 | IC50 | 3 | — | |
XZRCQWLPMXFGHE
|
6.5 | IC50 | 2 | — | |
KIMPACVVSQUMHL
|
6.5 | IC50 | 2 | — | |
GJJIICZAOJXOEJ
|
6.4 | IC50 | 2 | — | |
MWPKIJXVHHDLCZ
|
6.4 | IC50 | 2 | — | |
PCAWJIMDNGAMRA
|
6.4 | IC50 | 2 | — | |
RFKWWUGSOVDNFF
|
6.4 | IC50 | 2 | — | |
RMIJZTKTCJJVSA
|
6.3 | IC50 | 4 | — | |
HTTRFYNWHOXUPE
|
6.3 | IC50 | 3 | — | |
UOHKZMQXEJGUES
|
6.3 | IC50 | 4 | — |