Target Details
| UniProt AC | Q3Y6Q3 |
|---|---|
| Gene Symbol | blaVIM-2 |
| Protein Name | beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00753 (Lactamase_B) |
Summary
- Multi-target molecules 195
- Clinical molecules 0
- Avg pChEMBL 8.32
Active Molecules (195)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VDPWNHWRQQGIKF
|
7.8 | IC50 | 4 | — | |
DRIYJHIYAVHSCX
|
7.8 | IC50 | 4 | — | |
VGPOFZWUOHUAIP
|
7.8 | IC50 | 4 | — | |
YLRBRXDULGVRLL
|
7.8 | IC50 | 4 | — | |
AQWLIEJZSUSEDO
|
7.7 | IC50 | 4 | — | |
YLRBRXDULGVRLL
|
7.7 | IC50 | 4 | — | |
FVIOJUCTZRHDGE
|
7.7 | IC50 | 4 | — | |
OLXIFPYVDJEZDB
|
7.7 | IC50 | 4 | — | |
MSVXZGJHOFGLIG
|
7.7 | IC50 | 4 | — | |
YFUQHFWRSXGVPJ
|
7.6 | IC50 | 4 | — | |
IWMVHXGWCLSFTP
|
7.6 | IC50 | 4 | — | |
FQTKUOCDOGMYJK
|
7.6 | IC50 | 4 | — | |
PIPXFQLRUXMROV
|
7.6 | IC50 | 4 | — | |
RCVMXPMKZJWOML
|
7.6 | IC50 | 4 | — | |
OLGLXMCVCKKFMI
|
7.6 | IC50 | 4 | — | |
UXSBAEMCOIKVLS
|
7.6 | IC50 | 4 | — | |
IOBTYEBMEGZPSK
|
7.5 | IC50 | 4 | — | |
MXQBZELROZONIY
|
7.5 | IC50 | 4 | — | |
NVQTXRWKJYZJDM
|
7.5 | IC50 | 4 | — | |
ZLYBTODPVNLVES
|
7.4 | IC50 | 4 | — | |
IOBTYEBMEGZPSK
|
7.4 | IC50 | 4 | — | |
UTOBUGKFFQUTRB
|
7.4 | IC50 | 4 | — | |
PWGSAQYLORLIHN
|
7.3 | IC50 | 4 | — | |
ONLBWPOICXKPSH
|
7.3 | IC50 | 4 | — | |
UTPIDVLKEZUUCG
|
7.3 | IC50 | 4 | — | |
HCJUQKWZCHQJOX
|
7.3 | IC50 | 4 | — | |
MXQBZELROZONIY
|
7.3 | IC50 | 4 | — | |
AFTHORGZJFQNNK
|
7.2 | IC50 | 4 | — | |
XSTWRGDUYBPYCD
|
7.2 | IC50 | 4 | — | |
JBHZAUMQRROMLH
|
7.2 | IC50 | 4 | — | |
NTTWAYFZLWWMJH
|
7.2 | IC50 | 4 | — | |
GEFNYGUKJDHWHO
|
7.2 | IC50 | 4 | — | |
HWSQZBUPOYECIV
|
7.2 | IC50 | 4 | — | |
VKCKVSVYAJFTOH
|
7.2 | IC50 | 4 | — | |
MQFHAIUPLNBZFQ
|
7.1 | IC50 | 4 | — | |
WRTSDSXKEDBYNQ
|
6.9 | IC50 | 4 | — | |
PYSNWBGMHBFUBK
|
6.9 | IC50 | 4 | — | |
MQFHAIUPLNBZFQ
|
6.9 | IC50 | 4 | — | |
MPYHDNBHSKJGIR
|
6.8 | IC50 | 4 | — | |
GMNFCGZIQWNMMI
|
6.8 | IC50 | 4 | — | |
KDWPBDRWGSBBOS
|
6.7 | IC50 | 4 | — | |
NOKSEJLLZNSRQL
|
6.7 | IC50 | 4 | — | |
UMGGHKSXOCRGDE
|
6.7 | IC50 | 4 | — | |
UMGGHKSXOCRGDE
|
6.7 | IC50 | 4 | — | |
FXWFQAQXUDVIOS
|
6.7 | IC50 | 2 | — |