Target Details
| UniProt AC | Q388H8 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Glycylpeptide N-tetradecanoyltransferase |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01233 (NMT) PF02799 (NMT_C) |
Summary
- Multi-target molecules 275
- Clinical molecules 0
- Avg pChEMBL 8.03
Active Molecules (275)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LASGLELWXDVEQS
|
7.2 | IC50 | 2 | — | |
RRRIWYHXHUSTIG
|
7.2 | IC50 | 2 | — | |
JFVLKGVMXSZQKG
|
7.1 | IC50 | 2 | — | |
NSUPCQAJJZARPV
|
7.1 | IC50 | 2 | — | |
FZYMHWHBQLIJMR
|
7.1 | IC50 | 2 | — | |
SFBXFQFPPYDGMM
|
7.0 | IC50 | 2 | — | |
LHSFUTANKJPACJ
|
7.0 | IC50 | 2 | — | |
QOZMNUSRFBCGER
|
7.0 | IC50 | 2 | — | |
UZODOWRCBAMZPB
|
7.0 | IC50 | 3 | — | |
QWIODJSFIGQCMC
|
6.9 | IC50 | 2 | — | |
XZMZQDSXMWEWRG
|
6.9 | IC50 | 2 | — | |
YLYZSKPIJSILNO
|
6.8 | IC50 | 2 | — | |
UGQFKADYGVUGAY
|
6.8 | IC50 | 2 | — | |
OOAAJIDBDSUGSI
|
6.7 | IC50 | 2 | — | |
GZQJPTFJBDYKRV
|
6.7 | IC50 | 2 | — | |
AEYDRYLRVPXMRA
|
6.6 | IC50 | 2 | — | |
NJJQYISAKGZXAK
|
6.6 | IC50 | 2 | — | |
BAFTUTHSLRPADF
|
6.5 | IC50 | 2 | — | |
YYKHCFJYJZPKBK
|
6.5 | IC50 | 2 | — | |
BFZDMJJMYCHDIS
|
6.5 | IC50 | 2 | — | |
DDBJZLLZHMCDNB
|
6.5 | IC50 | 2 | — | |
HOIAFTVGAXSASA
|
6.4 | IC50 | 2 | — | |
CYUQRIULGOQGMA
|
6.4 | IC50 | 2 | — | |
PPRLWPOJFJTUNF
|
6.4 | IC50 | 2 | — | |
GQRWEJRYCBEXLY
|
6.2 | IC50 | 3 | — |