Target Details
| UniProt AC | Q388H8 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Glycylpeptide N-tetradecanoyltransferase |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01233 (NMT) PF02799 (NMT_C) |
Summary
- Multi-target molecules 275
- Clinical molecules 0
- Avg pChEMBL 8.03
Active Molecules (275)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DEZPLYCROJUSIB
|
7.7 | IC50 | 2 | — | |
HBWIVMZBEWFYKR
|
7.7 | IC50 | 2 | — | |
IXHQESXLKWPGHT
|
7.7 | IC50 | 3 | — | |
JQFOPXWJVQBOHK
|
7.7 | IC50 | 2 | — | |
ORJWGZRIGCSMHL
|
7.7 | IC50 | 3 | — | |
PQKLUVZCJZESDA
|
7.7 | IC50 | 3 | — | |
PSFHJBSFJDKCAK
|
7.7 | IC50 | 2 | — | |
SBZXVHLUNLYOOK
|
7.7 | IC50 | 2 | — | |
UZFFELQGDRFCKR
|
7.7 | IC50 | 2 | — | |
YTDRAOCSUIGLLJ
|
7.7 | IC50 | 3 | — | |
ZUZDCZMPAFAPSB
|
7.7 | IC50 | 3 | — | |
LSYBPIHGYXTNNH
|
7.6 | IC50 | 2 | — | |
VBGRETOBFIJKLG
|
7.6 | IC50 | 3 | — | |
XBGMDBGRBPVSAX
|
7.6 | IC50 | 3 | — | |
XSTSGMMNZAHGMW
|
7.6 | IC50 | 2 | — | |
HMTBKFYVOUJOGR
|
7.6 | IC50 | 2 | — | |
LLGNWULJKGEJSB
|
7.6 | IC50 | 2 | — | |
UEIHUROJPODEIZ
|
7.6 | IC50 | 3 | — | |
FFLACBJRLSONFM
|
7.6 | IC50 | 2 | — | |
NKPDOAKEBATUJP
|
7.6 | IC50 | 2 | — | |
RSFRJVKGQDTUAK
|
7.6 | IC50 | 3 | — | |
SURBAZXZJBJBJE
|
7.6 | IC50 | 2 | — | |
WSIAHLMGTALVDF
|
7.6 | IC50 | 2 | — | |
FGUZNVABRLKYEA
|
7.6 | IC50 | 3 | — | |
XJRSVURAWNRILV
|
7.6 | IC50 | 2 | — | |
NJADNIHZRBIIPB
|
7.6 | IC50 | 2 | — | |
WCZZAEZMIYIBTO
|
7.6 | IC50 | 2 | — | |
KSOHHJIWNDBIBO
|
7.5 | IC50 | 3 | — | |
PIHLQGWRCBUZIG
|
7.5 | IC50 | 2 | — | |
PRHLEXOVXVVUTM
|
7.5 | IC50 | 2 | — | |
UNOPBMXWYOSHGR
|
7.5 | IC50 | 2 | — | |
RPRVKMUKWQSFNP
|
7.5 | IC50 | 2 | — | |
WTWWPGQXKZXTQZ
|
7.5 | IC50 | 2 | — | |
ZLYXHAOYNACFLW
|
7.5 | IC50 | 2 | — | |
FFAHLLLCFOZVKL
|
7.5 | IC50 | 3 | — | |
SRVFWHXCZNTXTE
|
7.5 | IC50 | 3 | — | |
KJYPQUVUQWNMBI
|
7.5 | IC50 | 2 | — | |
LJJGCJROORPKCL
|
7.5 | IC50 | 2 | — | |
AVJKPNVHHCPBBW
|
7.4 | IC50 | 2 | — | |
QPIKSBVPHZNDOT
|
7.4 | IC50 | 3 | — | |
ZTIINHYISLWHNP
|
7.4 | IC50 | 2 | — | |
PQQYOZCMTKKSCS
|
7.4 | IC50 | 3 | — | |
YHCXRRMADSZIKJ
|
7.4 | IC50 | 3 | — | |
DXHKBDSGLAQZQY
|
7.3 | IC50 | 2 | — | |
JDDSAFSVBYQZKA
|
7.3 | IC50 | 2 | — | |
CLPBYHRNHCSBMR
|
7.3 | IC50 | 2 | — | |
RIYSPSXCDSEHMF
|
7.3 | IC50 | 2 | — | |
VAVJZHPOWKLYPG
|
7.3 | IC50 | 2 | — | |
XAWXGCBGDUJIJQ
|
7.3 | IC50 | 2 | — | |
MXPLBMZLFCIDHK
|
7.2 | IC50 | 2 | — |