Target Details
| UniProt AC | Q388H8 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Glycylpeptide N-tetradecanoyltransferase |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01233 (NMT) PF02799 (NMT_C) |
Summary
- Multi-target molecules 275
- Clinical molecules 0
- Avg pChEMBL 8.03
Active Molecules (275)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KMLSXJXNKKFPKB
|
8.1 | IC50 | 2 | — | |
MXDDYLKQWLNZOY
|
8.1 | IC50 | 2 | — | |
NNHIDDRNWJDOEK
|
8.1 | IC50 | 2 | — | |
QNDFBKGYIURDQZ
|
8.1 | IC50 | 2 | — | |
UZTUAUSVPXXHJG
|
8.1 | IC50 | 2 | — | |
ANEWXSRBOCZFRI
|
8.0 | IC50 | 2 | — | |
AUJGIZCNTFTZBQ
|
8.0 | IC50 | 2 | — | |
BTVULWWTNOUPPS
|
8.0 | IC50 | 2 | — | |
CRTSZBKSKNZCRS
|
8.0 | IC50 | 2 | — | |
DXXLBIFNGOCDOY
|
8.0 | IC50 | 2 | — | |
FHFKEHHLTWJRPV
|
8.0 | IC50 | 2 | — | |
FHLDEMLNIBTAGL
|
8.0 | IC50 | 3 | — | |
HAUGBCQQUOZSGH
|
8.0 | IC50 | 3 | — | |
HQHKSPQNNHMQTF
|
8.0 | IC50 | 3 | — | |
MATZARIBUNIWAK
|
8.0 | IC50 | 2 | — | |
NZJYJEBHJWAERL
|
8.0 | IC50 | 3 | — | |
TURQXTWKTXVDRW
|
8.0 | IC50 | 3 | — | |
TWZBEFAJLNTVPQ
|
8.0 | IC50 | 2 | — | |
XQFFEELKXUEKNR
|
8.0 | IC50 | 2 | — | |
XSONDNGKIAFWKK
|
8.0 | IC50 | 3 | — | |
YHOXDBJXAHZWCB
|
8.0 | IC50 | 2 | — | |
YKEDODVDSKYZBX
|
8.0 | IC50 | 2 | — | |
AJMGORHICVNZCC
|
8.0 | IC50 | 2 | — | |
BXFJLEZBOQBSPZ
|
8.0 | IC50 | 2 | — | |
FLCLHXMTMSHLQL
|
8.0 | IC50 | 2 | — | |
HBWNPNNLURLAIL
|
8.0 | IC50 | 2 | — | |
JAFYJORFMJAJBJ
|
8.0 | IC50 | 2 | — | |
MZECZFBGNUSGHF
|
8.0 | IC50 | 3 | — | |
PUVYTKKSEYNATO
|
8.0 | IC50 | 3 | — | |
YNZKRPJYTPZVOL
|
8.0 | IC50 | 2 | — | |
MONXKKKPSCPMRY
|
7.9 | IC50 | 2 | — | |
XJHUAHFZFJZMEE
|
7.9 | IC50 | 3 | — | |
GWKJWTPHSUXVCQ
|
7.9 | IC50 | 3 | — | |
YNMQWEFADPDXOL
|
7.8 | IC50 | 2 | — | |
ZGJHCUFFNQSMLI
|
7.8 | IC50 | 2 | — | |
GLLAAKIAMHKWQW
|
7.8 | IC50 | 3 | — | |
JPEQRKSUSLNASS
|
7.8 | IC50 | 3 | — | |
KZOYFHCJPGAJSW
|
7.8 | IC50 | 2 | — | |
MLQKDZOPUTYQGI
|
7.8 | IC50 | 2 | — | |
MUYWJBCCUVIPEV
|
7.8 | IC50 | 2 | — | |
OYNUBGTVBHOARA
|
7.8 | IC50 | 3 | — | |
TZBWLYPEOZFCKQ
|
7.8 | IC50 | 3 | — | |
XHOICLITTSTOPW
|
7.8 | IC50 | 2 | — | |
YFGXMQPXBQFQFQ
|
7.8 | IC50 | 2 | — | |
YVEXYAHGKCDEDN
|
7.8 | IC50 | 2 | — | |
XPWMJDXQGVZINH
|
7.8 | IC50 | 2 | — | |
GMNBTYGGCFCEHH
|
7.7 | IC50 | 3 | — | |
OTKMKBYGZQEUCC
|
7.7 | IC50 | 2 | — | |
VXNRXMGFBZVSJE
|
7.7 | IC50 | 2 | — | |
AGAPYTXFHCVDOQ
|
7.7 | IC50 | 2 | — |