Target Details
| UniProt AC | Q388H8 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Glycylpeptide N-tetradecanoyltransferase |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01233 (NMT) PF02799 (NMT_C) |
Summary
- Multi-target molecules 275
- Clinical molecules 0
- Avg pChEMBL 8.03
Active Molecules (275)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RKOABBUIRPYUAI
|
8.3 | IC50 | 2 | — | |
RNPIDPYYMUAVOZ
|
8.3 | IC50 | 2 | — | |
SEWQUULKELVECC
|
8.3 | IC50 | 2 | — | |
UMNGGVIIACWGNS
|
8.3 | IC50 | 2 | — | |
UVNZCVCPVURJHB
|
8.3 | IC50 | 2 | — | |
XANRCBWVKKVBOO
|
8.3 | IC50 | 3 | — | |
YJEDXBAVBHENKZ
|
8.3 | IC50 | 3 | — | |
AAUAFACIDYZGEN
|
8.2 | IC50 | 2 | — | |
AXUBNCKMKZTABP
|
8.2 | IC50 | 2 | — | |
CSPZQLIFXLIZAK
|
8.2 | IC50 | 3 | — | |
CTMRLURCRPZWBC
|
8.2 | IC50 | 3 | — | |
GMUQZULJZPZDRX
|
8.2 | IC50 | 2 | — | |
GNAUPOYUMUICBI
|
8.2 | IC50 | 3 | — | |
GRIZOICIXKRPIW
|
8.2 | IC50 | 3 | — | |
GUUDXDDOCWFTTL
|
8.2 | IC50 | 3 | — | |
HDXUATGUPZIGQP
|
8.2 | IC50 | 3 | — | |
HGAYHFOSEPDKPB
|
8.2 | IC50 | 2 | — | |
HRIXKKKRPHAAHK
|
8.2 | IC50 | 2 | — | |
ISOHWQXZGGNZKD
|
8.2 | IC50 | 2 | — | |
JCRQMWNGBUKXGD
|
8.2 | IC50 | 2 | — | |
JOUYDSVGXQRBPJ
|
8.2 | IC50 | 2 | — | |
MCEPYCPGZCPZQP
|
8.2 | IC50 | 2 | — | |
QVIGMASJSNWACY
|
8.2 | IC50 | 2 | — | |
RNBFWTPWSZZQMU
|
8.2 | IC50 | 2 | — | |
RTINSZYNDQPWSQ
|
8.2 | IC50 | 2 | — | |
SDTSVFNDBKQQQK
|
8.2 | IC50 | 3 | — | |
SQANARMSVUDZMB
|
8.2 | IC50 | 2 | — | |
TZGPVDMUGSMSTC
|
8.2 | IC50 | 2 | — | |
UBVLCBYJQLFVFT
|
8.2 | IC50 | 3 | — | |
VRBWPVWCIKKZEE
|
8.2 | IC50 | 2 | — | |
XKTNORGLMOOWAW
|
8.2 | IC50 | 2 | — | |
ZHBYGCKXGZISGA
|
8.2 | IC50 | 3 | — | |
ZZOMCUCZBJYMFA
|
8.2 | IC50 | 3 | — | |
ZZTPQQDXNJIJDB
|
8.2 | IC50 | 2 | — | |
DUUJIVZHYHCUKH
|
8.2 | IC50 | 2 | — | |
FKPKWRUZTWMINC
|
8.2 | IC50 | 2 | — | |
SGBQYQYDOKFCCS
|
8.2 | IC50 | 2 | — | |
VKVWILVVPXWBBP
|
8.2 | IC50 | 2 | — | |
WJEWMROJRZNDER
|
8.2 | IC50 | 2 | — | |
ZDOBVZZUCJJARZ
|
8.2 | IC50 | 2 | — | |
CPGZQBLXUHLONL
|
8.1 | IC50 | 2 | — | |
KPIUEPFVQHJKKR
|
8.1 | IC50 | 2 | — | |
MCBKFGPFRLYVIY
|
8.1 | IC50 | 2 | — | |
MTTYRLJXLWCQDU
|
8.1 | IC50 | 2 | — | |
MYSVDRKDBVTMJS
|
8.1 | IC50 | 2 | — | |
OOJBGWHNVNUTAW
|
8.1 | IC50 | 2 | — | |
VUJFBIQRCIUELB
|
8.1 | IC50 | 2 | — | |
ZOZYUQRKCVHRSB
|
8.1 | IC50 | 2 | — | |
DPRQAJSYCBYKDM
|
8.1 | IC50 | 2 | — | |
HSZRKOPMCINGBW
|
8.1 | IC50 | 2 | — |