Target Details
| UniProt AC | Q388H8 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Glycylpeptide N-tetradecanoyltransferase |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01233 (NMT) PF02799 (NMT_C) |
Summary
- Multi-target molecules 275
- Clinical molecules 0
- Avg pChEMBL 8.03
Active Molecules (275)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PLFXFPSZSLXQFL
|
8.5 | IC50 | 2 | — | |
PSMKGWAJXXDMRQ
|
8.5 | IC50 | 2 | — | |
QCMWJZZSCGOICB
|
8.5 | IC50 | 2 | — | |
QUOZSEHFMIATJW
|
8.5 | IC50 | 2 | — | |
REQUPDWBGITKAD
|
8.5 | IC50 | 2 | — | |
SWIZEMUQBPMLLW
|
8.5 | IC50 | 2 | — | |
UDGAVHUQIJVNHW
|
8.5 | IC50 | 2 | — | |
USALZGZGDFVTMX
|
8.5 | IC50 | 2 | — | |
VFSWJCSYVNBVSH
|
8.5 | IC50 | 2 | — | |
VGAIOTAXVWWJSW
|
8.5 | IC50 | 2 | — | |
VRZRGCVCKRCCLG
|
8.5 | IC50 | 2 | — | |
WZELAXINRXHZED
|
8.5 | IC50 | 2 | — | |
XEIMOGDDPRSYCR
|
8.5 | IC50 | 3 | — | |
XISLEJQCQIHTJT
|
8.5 | IC50 | 3 | — | |
YFWRJBGGRRIPTL
|
8.5 | IC50 | 2 | — | |
YMLFRSAHQNBEFS
|
8.5 | IC50 | 3 | — | |
YOJJQIDWBPPINE
|
8.5 | IC50 | 2 | — | |
YXVLLUQQJCRYSH
|
8.5 | IC50 | 2 | — | |
ZTCYDOMZBSOFPS
|
8.5 | IC50 | 2 | — | |
AJJUYNDFYWJVLC
|
8.4 | IC50 | 2 | — | |
FGWVXNIUFGLPRT
|
8.4 | IC50 | 3 | — | |
FSQFLTMLOZTAHB
|
8.4 | IC50 | 3 | — | |
FUWZRSVKKPXLIY
|
8.4 | IC50 | 3 | — | |
FYNYUDZLWFNZDV
|
8.4 | IC50 | 2 | — | |
IHJXCDLKNQEACS
|
8.4 | IC50 | 2 | — | |
IZKLXFJCDDXKPK
|
8.4 | IC50 | 2 | — | |
JJWNQGUDAZAITN
|
8.4 | IC50 | 2 | — | |
JSDZMSHSNXIWAC
|
8.4 | IC50 | 2 | — | |
KKALBIRLEONXKX
|
8.4 | IC50 | 3 | — | |
POTVFFXGRINLJD
|
8.4 | IC50 | 3 | — | |
PZIZCUMFALUOSC
|
8.4 | IC50 | 3 | — | |
QWBLERXEOLMUOE
|
8.4 | IC50 | 2 | — | |
RPZBHCIXTUDXGC
|
8.4 | IC50 | 3 | — | |
RSJADYGJFBJVKA
|
8.4 | IC50 | 2 | — | |
TWAIRZOVHJSHLQ
|
8.4 | IC50 | 2 | — | |
XVBSQNJZFGCFGT
|
8.4 | IC50 | 2 | — | |
XXKYMVWKLNFAHM
|
8.4 | IC50 | 2 | — | |
YQXVXYCNCZVVTG
|
8.4 | IC50 | 2 | — | |
ZJRMILCNIXBELO
|
8.4 | IC50 | 2 | — | |
AFNFIUZWTROPRZ
|
8.3 | IC50 | 2 | — | |
CGOWTXICZRDOFE
|
8.3 | IC50 | 2 | — | |
GROWGBVQGVDZRY
|
8.3 | IC50 | 2 | — | |
HGSRZOMBGXHVBF
|
8.3 | IC50 | 2 | — | |
IFDWZFPOQYAVFV
|
8.3 | IC50 | 3 | — | |
IYIKJWZFZWCRRP
|
8.3 | IC50 | 2 | — | |
KUYYPLKQMRSAHE
|
8.3 | IC50 | 2 | — | |
LPKLLYMRKISNCT
|
8.3 | IC50 | 2 | — | |
OLYYMDOJYFCFQN
|
8.3 | IC50 | 2 | — | |
PFWXHLNTKMHYOA
|
8.3 | IC50 | 3 | — | |
QDMPIQAZIKQCBE
|
8.3 | IC50 | 2 | — |