Target Details
| UniProt AC | Q388H8 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Glycylpeptide N-tetradecanoyltransferase |
| Organism | Trypanosoma brucei brucei (strain 927/4 GUTat10.1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01233 (NMT) PF02799 (NMT_C) |
Summary
- Multi-target molecules 275
- Clinical molecules 0
- Avg pChEMBL 8.03
Active Molecules (275)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BWKFDXGUFBWTCJ
|
9.0 | IC50 | 2 | — | |
DJAXIJFJXFFZSS
|
9.0 | IC50 | 2 | — | |
DSMKXBKHYODZJE
|
9.0 | IC50 | 2 | — | |
FNWCLKCMEUSKDI
|
9.0 | IC50 | 2 | — | |
FZVYQGHXJJDJEN
|
9.0 | IC50 | 2 | — | |
HCTLYQUKCDMZSK
|
9.0 | IC50 | 2 | — | |
MCLKNJADSXFFOA
|
9.0 | IC50 | 2 | — | |
PGZNGUIJEXFPJV
|
9.0 | IC50 | 2 | — | |
QNVZUWYJYIDRAI
|
9.0 | IC50 | 2 | — | |
WKTSLVQYGBHNRV
|
9.0 | IC50 | 2 | — | |
XMBSZPZJLPTFMV
|
9.0 | IC50 | 4 | — | |
ZRLPRQRWRDLYGQ
|
9.0 | IC50 | 2 | — | |
CJBFCFNKTFJGHD
|
8.7 | IC50 | 2 | — | |
HLJCVRXGZMOFDS
|
8.7 | IC50 | 4 | — | |
IACHGHVEEMFILS
|
8.7 | IC50 | 3 | — | |
JEXUGPIZWWTQHG
|
8.7 | IC50 | 3 | — | |
JHFMAYRHBZNEBV
|
8.7 | IC50 | 3 | — | |
JIXHFDPLDUQICU
|
8.7 | IC50 | 2 | — | |
JOAOLNUHUPTOJL
|
8.7 | IC50 | 2 | — | |
KZIRIBCVSGVRMY
|
8.7 | IC50 | 2 | — | |
LFUKSJMPHXRAHE
|
8.7 | IC50 | 3 | — | |
NWHUXUSJWDZLAZ
|
8.7 | IC50 | 2 | — | |
PPTHDMWUXYOQCC
|
8.7 | IC50 | 3 | — | |
QJZGKBFXCUBQLI
|
8.7 | IC50 | 2 | — | |
RAHQJHPEIGTWAB
|
8.7 | IC50 | 2 | — | |
RYJPWHHWIOKQFO
|
8.7 | IC50 | 3 | — | |
UGQSROIUKTXJQO
|
8.7 | IC50 | 3 | — | |
VHJREOZNHURPGO
|
8.7 | IC50 | 2 | — | |
WKXJMUPONLJJAH
|
8.7 | IC50 | 2 | — | |
ANDYEVOGBRSBAM
|
8.5 | IC50 | 2 | — | |
BOHQHSGCHQSRHG
|
8.5 | IC50 | 2 | — | |
COJPRJCSLJKNNT
|
8.5 | IC50 | 3 | — | |
DDXKXYFTXRXBNA
|
8.5 | IC50 | 2 | — | |
DRBQXWGZAGDOEL
|
8.5 | IC50 | 2 | — | |
DVTQRRNJAIULRN
|
8.5 | IC50 | 3 | — | |
DYBVVKGMMMWRHW
|
8.5 | IC50 | 2 | — | |
FGXSOXXSWXJIQM
|
8.5 | IC50 | 2 | — | |
GASUPAQGJGLLGM
|
8.5 | IC50 | 3 | — | |
GHEOOJQNTOZPOE
|
8.5 | IC50 | 2 | — | |
GVYHLYWBDITGOO
|
8.5 | IC50 | 3 | — | |
KFZNUMAAQRKTIR
|
8.5 | IC50 | 3 | — | |
KGUSVAQCTAVWAD
|
8.5 | IC50 | 3 | — | |
LKMRBDPAMYFBMF
|
8.5 | IC50 | 2 | — | |
MOPOVPPQSBKKPE
|
8.5 | IC50 | 2 | — | |
NCFHKHWPNGZJEO
|
8.5 | IC50 | 3 | — | |
NYWHVKZUMUDVFT
|
8.5 | IC50 | 2 | — | |
OYCYNVBHMJSUKL
|
8.5 | IC50 | 2 | — | |
OZDFQTLYOJBXDX
|
8.5 | IC50 | 2 | — | |
PGRFAUBJFXTXLR
|
8.5 | IC50 | 3 | — | |
PINSRGHFBUSSTB
|
8.5 | IC50 | 3 | — |