Target Details
| UniProt AC | Q32MK0 |
|---|---|
| Gene Symbol | MYLK3 |
| Protein Name | Myosin light chain kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 27
- Clinical molecules 11
- Avg pChEMBL 6.97
KEGG Pathways (10)
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PIQCTGMSNWUMAF
|
8.7 | Kd | 137 | Yes | |
YYLKKYCXAOBSRM
|
8.4 | Kd | 191 | — | |
UIARLYUEJFELEN
|
7.9 | Kd | 289 | Yes | |
GCIKSSRWRFVXBI
|
7.8 | Kd | 109 | Yes | |
WINHZLLDWRZWRT
|
7.6 | Kd | 201 | Yes | |
YFNWWNRZJGMDBR
|
7.5 | Kd | 35 | — | |
CTNPALGJUAXMMC
|
7.4 | Kd | 151 | — | |
GUBJNPWVIUFSTR
|
7.4 | Kd | 103 | — | |
KOZFSFOOLUUIGY
|
7.0 | Kd | 88 | Yes | |
QTBWCSQGBMPECM
|
7.0 | Kd | 21 | Yes | |
RYYNGWLOYLRZLK
|
7.0 | Kd | 45 | — | |
XZXHXSATPCNXJR
|
7.0 | Kd | 165 | Yes | |
LOLPPWBBNUVNQZ
|
6.9 | Kd | 97 | Yes | |
HKSZLNNOFSGOKW
|
6.8 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
6.8 | Kd | 213 | — | |
VAARYSWULJUGST
|
6.8 | Kd | 119 | Yes | |
NXSJMRCTGYTSTK
|
6.8 | Kd | 200 | — | |
GMIZZEXBPRLVIV
|
6.7 | Kd | 6 | — | |
MWKSRKSEWLRPBL
|
6.5 | Kd | 1075 | — | |
AYCPARAPKDAOEN
|
6.5 | Kd | 73 | — | |
MFAQYJIYDMLAIM
|
6.4 | Kd | 130 | Yes | |
BPNUQXPIQBZCMR
|
6.4 | Kd | 83 | Yes | |
CVWXJKQAOSCOAB
|
6.4 | Kd | 35 | — | |
XDJCLCLBSGGNKS
|
6.3 | Kd | 21 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |