Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PQRRTYZMKUUTSQ
|
9.2 | IC50 | 4 | — | |
WNEHLMHMEYRECK
|
9.2 | IC50 | 4 | — | |
ZRPQKMDBBKACFK
|
9.2 | IC50 | 4 | — | |
UFZKDWACGLCXKW
|
9.2 | IC50 | 4 | — | |
QYMNHYZLJVXASV
|
9.2 | IC50 | 4 | — | |
HPURORKUCWKUFZ
|
9.2 | IC50 | 4 | — | |
HURUOGCXPHOTEQ
|
9.2 | IC50 | 4 | — | |
QFYYYMBQAPXZRF
|
9.2 | IC50 | 4 | — | |
PXYFMAZFKVHGCP
|
9.2 | IC50 | 4 | — | |
GLBQLNGOYWLSPB
|
9.1 | IC50 | 4 | — | |
GRGVOQXAHCJURA
|
9.1 | IC50 | 4 | — | |
LBJBSCVPRJVYAR
|
9.1 | IC50 | 4 | — | |
LQLKYWFVAIUUME
|
9.1 | IC50 | 4 | — | |
VTIMNZCVMMQWBP
|
9.1 | IC50 | 3 | — | |
ZRPQKMDBBKACFK
|
9.1 | IC50 | 3 | — | |
ZWPMTWURJWGRPP
|
9.1 | IC50 | 4 | — | |
VDJGSMHUOZCHIH
|
9.1 | IC50 | 4 | — | |
XXVBQYHIFYSDQC
|
9.1 | IC50 | 4 | — | |
DRKUCVWOBRAQJJ
|
9.1 | IC50 | 4 | — | |
AWFLVGLEZADZME
|
9.1 | IC50 | 4 | — | |
PMDPQFMJDBKWKX
|
9.1 | IC50 | 4 | — | |
XZEDAOVENNDOSA
|
9.1 | IC50 | 4 | — | |
FSBJMTPSCUKYHG
|
9.0 | IC50 | 4 | — | |
PMDPQFMJDBKWKX
|
9.0 | IC50 | 4 | — | |
SHVIQNRXTAJHCL
|
9.0 | IC50 | 4 | — | |
IHDWQPGJKYAEGB
|
9.0 | IC50 | 4 | — | |
YJLWZMRIPUTANI
|
9.0 | IC50 | 4 | — | |
BQDSHDWYJINFEE
|
9.0 | IC50 | 4 | — | |
NGXJGSGMLDIREA
|
9.0 | IC50 | 4 | — | |
XZEDAOVENNDOSA
|
9.0 | IC50 | 4 | — | |
QXJUVJZYKOFZPK
|
9.0 | IC50 | 4 | — | |
URIMKCJWSVIKRZ
|
9.0 | IC50 | 4 | — | |
AUDKQARKDIVADP
|
9.0 | IC50 | 4 | — | |
HFOJOTOEYNQQED
|
9.0 | IC50 | 4 | — | |
UMBJQXVDZMLNAG
|
9.0 | IC50 | 4 | — | |
AYUSQLJTKXUKDZ
|
8.9 | IC50 | 4 | — | |
SYSQZTFYEUUIMG
|
8.9 | IC50 | 4 | — | |
UTJPHSHUPFTYLW
|
8.9 | IC50 | 4 | — | |
ANTMOAIWXABXQH
|
8.9 | IC50 | 4 | — | |
PJDYNGJJKINRRX
|
8.9 | IC50 | 4 | — | |
UMHFRIKKMWUBNA
|
8.9 | IC50 | 4 | — | |
QDKBOVSCISEIKW
|
8.9 | IC50 | 4 | — | |
ASHSVVZOBGBBQZ
|
8.8 | IC50 | 4 | — | |
SVUZRMIRYAQATK
|
8.8 | IC50 | 4 | — | |
DZSRWIWGTYSZLQ
|
8.8 | IC50 | 4 | — | |
QSHBWYDCKYJNCO
|
8.8 | IC50 | 4 | — | |
UZDRIDPZPMGZOL
|
8.8 | IC50 | 4 | — | |
GGNOUJIQFPIIRP
|
8.8 | IC50 | 4 | — | |
GGNOUJIQFPIIRP
|
8.8 | IC50 | 4 | — | |
FFFYJIJMAQAFDJ
|
8.8 | IC50 | 4 | — |