Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UKNSUAZTZOWTCO
|
9.5 | IC50 | 4 | — | |
WWNJZLQOIDKOIT
|
9.5 | IC50 | 4 | — | |
KRUJLHIBOQDVQO
|
9.5 | IC50 | 3 | — | |
YLUNJCYDQAOVHO
|
9.4 | IC50 | 4 | — | |
FDGVFDRSCMPIBM
|
9.4 | IC50 | 4 | — | |
MXTWYAUYKBJDQV
|
9.4 | IC50 | 3 | — | |
IGKPYTKMVZOTKY
|
9.4 | IC50 | 4 | — | |
JMGDTOZRWTXGIB
|
9.4 | IC50 | 4 | — | |
RPFSQALYXQGHSI
|
9.4 | IC50 | 4 | — | |
UKBZTXIKOMESBJ
|
9.4 | IC50 | 4 | — | |
XJDUVCNADJGFCF
|
9.4 | IC50 | 4 | — | |
IQVSMXLKXITUHA
|
9.4 | IC50 | 4 | — | |
ZFUKHIWTVAISFP
|
9.4 | IC50 | 4 | — | |
JTQVEIOPHVMFAR
|
9.4 | IC50 | 4 | — | |
PYLGNAIHDHKRKU
|
9.4 | IC50 | 4 | — | |
VTCZVSYBKZUREZ
|
9.4 | IC50 | 4 | — | |
XMXWDQIXFXAIEG
|
9.4 | IC50 | 4 | — | |
YZXXIGRHLIBEIM
|
9.4 | IC50 | 4 | — | |
HURUOGCXPHOTEQ
|
9.4 | IC50 | 4 | — | |
SRWZJCQAFWBVNN
|
9.4 | IC50 | 4 | — | |
VADZVCWYZHWQOX
|
9.4 | IC50 | 4 | — | |
YZXXIGRHLIBEIM
|
9.4 | IC50 | 4 | — | |
COEMWBDMVJOSNX
|
9.3 | IC50 | 4 | — | |
FXKBDOWBFUHQLK
|
9.3 | IC50 | 4 | — | |
IGKPYTKMVZOTKY
|
9.3 | IC50 | 4 | — | |
UXNGUTOGQXUODT
|
9.3 | IC50 | 4 | — | |
VDGZDOXAAFBKEX
|
9.3 | IC50 | 4 | — | |
ADGAXIHGUNIVHL
|
9.3 | IC50 | 3 | — | |
VXBFUHKHJXONAB
|
9.3 | IC50 | 4 | — | |
CHZMHLGFIPQNHF
|
9.3 | IC50 | 4 | — | |
WGCIOOTXJABATI
|
9.3 | IC50 | 4 | — | |
ARBCOGFEJXLOLI
|
9.3 | IC50 | 4 | — | |
JRUSWFUCBJJDSX
|
9.3 | IC50 | 4 | — | |
KQHJVFYEQCPAAB
|
9.3 | IC50 | 4 | — | |
MOHHMIRAZDGHTA
|
9.3 | IC50 | 4 | — | |
PQRRTYZMKUUTSQ
|
9.3 | IC50 | 4 | — | |
SIWCWAWNBNHPRL
|
9.3 | IC50 | 4 | — | |
YRJUQGHTWWYHCP
|
9.3 | IC50 | 4 | — | |
YFZRDNDRLVDZJA
|
9.3 | IC50 | 4 | — | |
HNNSSWVDZVWCER
|
9.3 | IC50 | 4 | — | |
ZJHKDXMGXOZAKR
|
9.3 | IC50 | 4 | — | |
GYGNYDYNNRAFMQ
|
9.3 | IC50 | 4 | — | |
NUGIVIRZGIFIKC
|
9.3 | IC50 | 4 | — | |
BLGYKMGOMSKCTK
|
9.3 | IC50 | 4 | — | |
OZTGBIOQFYIWIA
|
9.3 | IC50 | 4 | — | |
YZUWHIDXKAVWBK
|
9.3 | IC50 | 4 | — | |
IOQCZQUVXNEXKO
|
9.2 | IC50 | 4 | — | |
LRODNFJRCKXACM
|
9.2 | IC50 | 4 | — | |
MHMCEJWETAYNFG
|
9.2 | IC50 | 4 | — | |
YFQVRYQHRYRIBR
|
9.2 | IC50 | 4 | — |