Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BTRCLHPJGPGTTQ
|
9.6 | IC50 | 4 | — | |
CRRHXDQIJGYZET
|
9.6 | IC50 | 4 | — | |
FTXGUAGAMDIGQY
|
9.6 | IC50 | 4 | — | |
NRGZZANDJWYHMJ
|
9.6 | IC50 | 3 | — | |
QCQUIPYGOWSNKA
|
9.6 | IC50 | 4 | — | |
QLPRLZKQKAZIAD
|
9.6 | IC50 | 4 | — | |
QVKQWKSQEZEBGV
|
9.6 | IC50 | 4 | — | |
XOQHYOIVBAXCRE
|
9.6 | IC50 | 4 | — | |
KBEFGPUEURSHSQ
|
9.6 | IC50 | 4 | — | |
RYFBXXBUFPDLOZ
|
9.6 | IC50 | 3 | — | |
CFQYUHDEIHGDPN
|
9.6 | IC50 | 4 | — | |
JMGDTOZRWTXGIB
|
9.6 | IC50 | 4 | — | |
OARACMMQYKDCQI
|
9.6 | IC50 | 4 | — | |
QCAQSGLKDSNCDV
|
9.6 | IC50 | 4 | — | |
SAKGTUDYUKGYQO
|
9.6 | IC50 | 4 | — | |
SGZFQFBJJXRGIS
|
9.6 | IC50 | 4 | — | |
DXXYBYNBBDJSNY
|
9.5 | IC50 | 4 | — | |
PHSIHADDWCLCLE
|
9.5 | IC50 | 4 | — | |
SBOAFHKVXFONAG
|
9.5 | IC50 | 4 | — | |
VQFVDKZCXCUSNA
|
9.5 | IC50 | 4 | — | |
JSSNYCYCQLWUEO
|
9.5 | IC50 | 4 | — | |
MQPNMUKUHJVESA
|
9.5 | IC50 | 4 | — | |
NUVVRDXSOKREQQ
|
9.5 | IC50 | 4 | — | |
ODMPCHPWIKBECJ
|
9.5 | IC50 | 4 | — | |
XONJRNLITDZUPT
|
9.5 | IC50 | 4 | — | |
DTEHDBCPEXVDDP
|
9.5 | IC50 | 4 | — | |
GAFUGIBXFLEVLZ
|
9.5 | IC50 | 4 | — | |
HIKFETGSIFPCHR
|
9.5 | IC50 | 4 | — | |
JEDUPUZDNZUVNK
|
9.5 | IC50 | 4 | — | |
KRUJLHIBOQDVQO
|
9.5 | IC50 | 4 | — | |
YRYJPVHXXMDXMA
|
9.5 | IC50 | 4 | — | |
ZULUBCFYHQEBJW
|
9.5 | IC50 | 4 | — | |
CONFNNPDLZWHGO
|
9.5 | IC50 | 4 | — | |
DFSHPCNEJBOKNO
|
9.5 | IC50 | 4 | — | |
IZVFPCAFESKVCW
|
9.5 | IC50 | 4 | — | |
VTCZVSYBKZUREZ
|
9.5 | IC50 | 4 | — | |
YHCLLRXKMQSION
|
9.5 | IC50 | 4 | — | |
CUPNOXUVTFMQBF
|
9.5 | IC50 | 4 | — | |
FBOXLDIWBOPBGH
|
9.5 | IC50 | 4 | — | |
FTCIEXDPNOJVHG
|
9.5 | IC50 | 4 | — | |
WTHMCCLQHZUJPX
|
9.5 | IC50 | 4 | — | |
ZJHKDXMGXOZAKR
|
9.5 | IC50 | 3 | — | |
CUPNOXUVTFMQBF
|
9.5 | IC50 | 3 | — | |
IRSQPGJWCQJGBA
|
9.5 | IC50 | 4 | — | |
JMGDTOZRWTXGIB
|
9.5 | IC50 | 4 | — | |
OEDGFHOVDDKFPY
|
9.5 | IC50 | 4 | — | |
USMNMZULIAYFEJ
|
9.5 | IC50 | 4 | — | |
YAFPNJUNYYCEJF
|
9.5 | IC50 | 4 | — | |
BKKUNWMBSWSMJT
|
9.5 | IC50 | 4 | — | |
PRVKGOPWBRUUTC
|
9.5 | IC50 | 3 | — |