Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DFEIOWJQIXAABN
|
9.7 | IC50 | 4 | — | |
HGICSZSMZDNVQQ
|
9.7 | IC50 | 4 | — | |
JHJTVOYFIGVQSN
|
9.7 | IC50 | 4 | — | |
KXELUNLBQPTQIB
|
9.7 | IC50 | 4 | — | |
CADODRJOFDTRLR
|
9.7 | IC50 | 4 | — | |
JSSNYCYCQLWUEO
|
9.7 | IC50 | 4 | — | |
KJCSBMYFBQKAEH
|
9.7 | IC50 | 4 | — | |
MWQOZPQHEVVWNU
|
9.7 | IC50 | 4 | — | |
VOUWZRKTKXPBRF
|
9.7 | IC50 | 4 | — | |
WMAUGRQDBDVUIO
|
9.7 | IC50 | 4 | — | |
XHSAXLCYFREUHS
|
9.7 | IC50 | 4 | — | |
CXSKGFQNMGEJNL
|
9.6 | IC50 | 4 | — | |
DSUJPDGATORSMZ
|
9.6 | IC50 | 4 | — | |
FBXDTPCRCZBDAX
|
9.6 | IC50 | 4 | — | |
VXBFUHKHJXONAB
|
9.6 | IC50 | 4 | — | |
BZSYHKGTTGQSDN
|
9.6 | IC50 | 4 | — | |
CUPNOXUVTFMQBF
|
9.6 | IC50 | 4 | — | |
CUZJLQPCENXUCT
|
9.6 | IC50 | 4 | — | |
FWQZETXDUPNNGK
|
9.6 | IC50 | 4 | — | |
INXQISMCTPPLKA
|
9.6 | IC50 | 4 | — | |
JIJWPANZXWZBEY
|
9.6 | IC50 | 4 | — | |
PUWJQTDZRWOSDD
|
9.6 | IC50 | 3 | — | |
SBOAFHKVXFONAG
|
9.6 | IC50 | 4 | — | |
XBTNMJXWTUCPMA
|
9.6 | IC50 | 4 | — | |
XSWVMWMRFVXDMM
|
9.6 | IC50 | 4 | — | |
YUFZAQCMPXKUOU
|
9.6 | IC50 | 4 | — | |
CSQYQNBGABBMEH
|
9.6 | IC50 | 4 | — | |
KZEKVTGPSJUAQG
|
9.6 | IC50 | 4 | — | |
QPZMHHDLQNWPAO
|
9.6 | IC50 | 4 | — | |
RRTXSFAFHOPSAU
|
9.6 | IC50 | 4 | — | |
SGZFQFBJJXRGIS
|
9.6 | IC50 | 4 | — | |
SRVMJNHIRBPMGD
|
9.6 | IC50 | 4 | — | |
SRWZJCQAFWBVNN
|
9.6 | IC50 | 4 | — | |
VOUWZRKTKXPBRF
|
9.6 | IC50 | 4 | — | |
ZOIGAFIIRTZXOR
|
9.6 | IC50 | 4 | — | |
FYFIFUQBONLCMI
|
9.6 | IC50 | 4 | — | |
HIKFETGSIFPCHR
|
9.6 | IC50 | 4 | — | |
JLNIEZHUHKZAPH
|
9.6 | IC50 | 4 | — | |
JTJBIUPVRAYOQB
|
9.6 | IC50 | 4 | — | |
LBUOPPLAHISZMY
|
9.6 | IC50 | 4 | — | |
PKHNATXKSLXAEY
|
9.6 | IC50 | 4 | — | |
YRYJPVHXXMDXMA
|
9.6 | IC50 | 4 | — | |
INXQISMCTPPLKA
|
9.6 | IC50 | 4 | — | |
JLDQAFWPTZLUPS
|
9.6 | IC50 | 4 | — | |
LITRKXUVXQDMIS
|
9.6 | IC50 | 4 | — | |
PQRRTYZMKUUTSQ
|
9.6 | IC50 | 4 | — | |
GXXINTLQYNYOCT
|
9.6 | IC50 | 4 | — | |
SHVIQNRXTAJHCL
|
9.6 | IC50 | 4 | — | |
VTIMNZCVMMQWBP
|
9.6 | IC50 | 4 | — | |
VVGDNPGVZIEQAP
|
9.6 | IC50 | 4 | — |