Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JLQLVMLCSVSHON
|
9.8 | IC50 | 4 | — | |
JMGDTOZRWTXGIB
|
9.8 | IC50 | 4 | — | |
SBKXCXIHIWLXOS
|
9.8 | IC50 | 4 | — | |
VICRGYUMXJXQAL
|
9.8 | IC50 | 4 | — | |
WWOWQFNSNPLLCR
|
9.8 | IC50 | 4 | — | |
XGFAJSGBLMHBHK
|
9.8 | IC50 | 4 | — | |
YQHBXQCEAXBCEQ
|
9.8 | IC50 | 4 | — | |
FZQGKUYDMKKPSR
|
9.8 | IC50 | 4 | — | |
GQMKFJFLZZHKEE
|
9.8 | IC50 | 4 | — | |
PQRRTYZMKUUTSQ
|
9.8 | IC50 | 4 | — | |
UELOJMHIIBZDFG
|
9.8 | IC50 | 4 | — | |
GINLASFWCXLJSB
|
9.8 | IC50 | 4 | — | |
REQDHYOMMZXOKJ
|
9.8 | IC50 | 4 | — | |
WKCXBSWUNFBPJA
|
9.8 | IC50 | 4 | — | |
FPDSKARHYNDHLY
|
9.8 | IC50 | 4 | — | |
GYGNYDYNNRAFMQ
|
9.8 | IC50 | 4 | — | |
JIJWPANZXWZBEY
|
9.8 | IC50 | 4 | — | |
JKAOOUXUHVNVNM
|
9.8 | IC50 | 4 | — | |
KCQQRBQSGGONSX
|
9.8 | IC50 | 4 | — | |
NEVMFJXLRZQHHL
|
9.8 | IC50 | 4 | — | |
XFNUOVGFHOBFAS
|
9.8 | IC50 | 4 | — | |
YZUWHIDXKAVWBK
|
9.8 | IC50 | 4 | — | |
AFJIDACMIUWLIM
|
9.8 | IC50 | 4 | — | |
BZRQYXDEDLYNGM
|
9.8 | IC50 | 4 | — | |
HEXNYHIYGROCAJ
|
9.8 | IC50 | 4 | — | |
MMMKNRDKALEWNQ
|
9.8 | IC50 | 4 | — | |
PFGLEWSOALRQSL
|
9.8 | IC50 | 4 | — | |
QSASZUPKWFJGDP
|
9.8 | IC50 | 4 | — | |
SAKGTUDYUKGYQO
|
9.8 | IC50 | 4 | — | |
YXLGKVLZNAGKOT
|
9.8 | IC50 | 4 | — | |
LETKBQVLHMERPP
|
9.8 | IC50 | 4 | — | |
MIAXLWJVTIMZHF
|
9.8 | IC50 | 4 | — | |
NJNPJGQDAFDHTB
|
9.8 | IC50 | 4 | — | |
SSSFMTDTKCJFRF
|
9.8 | IC50 | 4 | — | |
UQTMNFPUWSWOOK
|
9.8 | IC50 | 4 | — | |
VCZHTULROJWCDK
|
9.8 | IC50 | 4 | — | |
ZHEASBZRWARPLY
|
9.8 | IC50 | 4 | — | |
AZCKVKUWLPBOMP
|
9.7 | IC50 | 4 | — | |
BOWSJWYIIKQERX
|
9.7 | IC50 | 4 | — | |
DGBXDGANRYBJPM
|
9.7 | IC50 | 4 | — | |
DSYLPQWDXAPXNT
|
9.7 | IC50 | 4 | — | |
HGTMGNYFIGMTIZ
|
9.7 | IC50 | 4 | — | |
JIJWPANZXWZBEY
|
9.7 | IC50 | 4 | — | |
PKIKBIFPRCUBFS
|
9.7 | IC50 | 4 | — | |
QJGBZMFDMGHLPK
|
9.7 | IC50 | 4 | — | |
SZMQVONRDOVLLM
|
9.7 | IC50 | 4 | — | |
WGFTVTKLTQAKIN
|
9.7 | IC50 | 4 | — | |
WWFBADABYQJEOH
|
9.7 | IC50 | 4 | — | |
YHCLLRXKMQSION
|
9.7 | IC50 | 4 | — | |
YREYWLTWIWCHHP
|
9.7 | IC50 | 4 | — |