Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MDKTUBIZBKMCTP
|
9.9 | IC50 | 4 | — | |
MSMJGPZJICCOHZ
|
9.9 | IC50 | 4 | — | |
QCEPJZBJONEUOB
|
9.9 | IC50 | 4 | — | |
WEEHEDJDVSMSOI
|
9.9 | IC50 | 4 | — | |
AKCFPSXRYKMLQV
|
9.9 | IC50 | 4 | — | |
CQVYWECRQQVMBR
|
9.9 | IC50 | 4 | — | |
CWJKRRQBAPFZIH
|
9.9 | IC50 | 4 | — | |
DJSACFIVKUCITB
|
9.9 | IC50 | 4 | — | |
DUWAWPVUNJBRQD
|
9.9 | IC50 | 4 | — | |
GAQHWLUIEFDDDA
|
9.9 | IC50 | 4 | — | |
IHDWQPGJKYAEGB
|
9.9 | IC50 | 4 | — | |
IOZRHZRRSVGYHP
|
9.9 | IC50 | 4 | — | |
IOZRHZRRSVGYHP
|
9.9 | IC50 | 4 | — | |
KPPVDQNDBNNEFB
|
9.9 | IC50 | 4 | — | |
NNFCNZSFFWFISR
|
9.9 | IC50 | 4 | — | |
PDXARPUHKHFKLG
|
9.9 | IC50 | 4 | — | |
KQHZWEWCZJWCIF
|
9.9 | IC50 | 4 | — | |
MPKFPGZSQMILTQ
|
9.9 | IC50 | 5 | — | |
PULJZVSXVWZSIQ
|
9.9 | IC50 | 4 | — | |
SETGFHFOFNXULG
|
9.9 | IC50 | 4 | — | |
WEHSIJUBIMRXIV
|
9.9 | IC50 | 3 | — | |
FLIUGCCDOLARIN
|
9.9 | IC50 | 4 | — | |
TVOOVNFXLKCVSE
|
9.9 | IC50 | 4 | — | |
GDJXWHAPBJZDJG
|
9.8 | IC50 | 4 | — | |
IWTXQBNOWPLXHV
|
9.8 | IC50 | 4 | — | |
PYXMLVCFVAGROW
|
9.8 | IC50 | 4 | — | |
UQABAZIVOWVRHR
|
9.8 | IC50 | 4 | — | |
XQMXOQCDPKRVCW
|
9.8 | IC50 | 4 | — | |
ZHEASBZRWARPLY
|
9.8 | IC50 | 4 | — | |
BKJNWVSHORBYDI
|
9.8 | IC50 | 4 | — | |
DHHOUQGEQFJXDP
|
9.8 | IC50 | 4 | — | |
JBDBUJFWVODNTD
|
9.8 | IC50 | 4 | — | |
XUTLQVNLWMGEBG
|
9.8 | IC50 | 4 | — | |
CJGHWHVRPSCRKH
|
9.8 | IC50 | 4 | — | |
CYDKMYNWSJUBBJ
|
9.8 | IC50 | 4 | — | |
KCNOJKKSHLOHOR
|
9.8 | IC50 | 3 | — | |
KTHPBOABEUUPEP
|
9.8 | IC50 | 4 | — | |
RFVBSTIXVQLSRH
|
9.8 | IC50 | 4 | — | |
AEEHUJLNCWTCAO
|
9.8 | IC50 | 4 | — | |
IZBVNRDYZNDUQA
|
9.8 | IC50 | 4 | — | |
JNEHDYVJEYMSIB
|
9.8 | IC50 | 4 | — | |
JUDRIABXAXKJJO
|
9.8 | IC50 | 4 | — | |
NBQHXIGLUPQFLR
|
9.8 | IC50 | 4 | — | |
NDLQJZOEBQXRFC
|
9.8 | IC50 | 4 | — | |
TXXWCRQWLDPAJM
|
9.8 | IC50 | 4 | — | |
YUBFCSFQTYJUHP
|
9.8 | IC50 | 4 | — | |
HVZNGQAYECGPHO
|
9.8 | IC50 | 4 | — | |
LEJNHZRHSOULSO
|
9.8 | IC50 | 4 | — | |
MOMXDEZGVCWDGR
|
9.8 | IC50 | 4 | — | |
BZRQYXDEDLYNGM
|
9.8 | IC50 | 4 | — |