Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SSQJGJDTNDSZCF
|
10.0 | IC50 | 4 | — | |
VUOAFRFMPXVXJW
|
10.0 | IC50 | 4 | — | |
AVQUBGSNDSFZMU
|
10.0 | IC50 | 4 | — | |
LEJNHZRHSOULSO
|
10.0 | IC50 | 4 | — | |
MUHGOHRJHQLIJS
|
10.0 | IC50 | 4 | — | |
SEZAYZOWIOZWCF
|
10.0 | IC50 | 4 | — | |
XLRPXJWNTZKRLK
|
10.0 | IC50 | 3 | — | |
GZBHDBFPVJZAKJ
|
10.0 | IC50 | 4 | — | |
SLNRHOOIEOVENH
|
10.0 | IC50 | 4 | — | |
SXKLZDRFRIVRMH
|
10.0 | IC50 | 4 | — | |
UBSHWFYWCAQXGO
|
10.0 | IC50 | 4 | — | |
UJGPUAGSBLTGDV
|
10.0 | IC50 | 3 | — | |
ABAPJYDJVJVZSN
|
9.9 | IC50 | 4 | — | |
BNUKGEOODPQOPU
|
9.9 | IC50 | 4 | — | |
JBDBUJFWVODNTD
|
9.9 | IC50 | 4 | — | |
JZLLJZAPAPKAQY
|
9.9 | IC50 | 4 | — | |
PDXARPUHKHFKLG
|
9.9 | IC50 | 4 | — | |
PQOCNUYHZWCRFU
|
9.9 | IC50 | 4 | — | |
BSSOREZAYOZEAB
|
9.9 | IC50 | 4 | — | |
HLXWUESRDMZWKV
|
9.9 | IC50 | 4 | — | |
IIUCDOABIKQJOU
|
9.9 | IC50 | 4 | — | |
LVZHNFNNMLWQEX
|
9.9 | IC50 | 4 | — | |
NUVVRDXSOKREQQ
|
9.9 | IC50 | 4 | — | |
OARACMMQYKDCQI
|
9.9 | IC50 | 4 | — | |
RJFSUXPNRYMHRA
|
9.9 | IC50 | 4 | — | |
SYSQZTFYEUUIMG
|
9.9 | IC50 | 4 | — | |
WLWWKCMOTWEMIB
|
9.9 | IC50 | 4 | — | |
XFNUOVGFHOBFAS
|
9.9 | IC50 | 4 | — | |
NJKDZCGDZKEPQP
|
9.9 | IC50 | 4 | — | |
UFZKDWACGLCXKW
|
9.9 | IC50 | 4 | — | |
UYCSHUDHNCMRBK
|
9.9 | IC50 | 4 | — | |
BYOIHNHEFHNPER
|
9.9 | IC50 | 4 | — | |
IAQFFDQRSKBBQD
|
9.9 | IC50 | 4 | — | |
NBQHXIGLUPQFLR
|
9.9 | IC50 | 4 | — | |
NGJUIXRTMZQSAK
|
9.9 | IC50 | 4 | — | |
OXTCIOGTSMOFPV
|
9.9 | IC50 | 4 | — | |
OYHMXKMDUJOANP
|
9.9 | IC50 | 4 | — | |
UPTYLORMCUHQQZ
|
9.9 | IC50 | 4 | — | |
YMUHBVLKRVQAKO
|
9.9 | IC50 | 4 | — | |
ASZICAZGNIKFEG
|
9.9 | IC50 | 4 | — | |
JIGOZOQZFQGGRB
|
9.9 | IC50 | 4 | — | |
SXKLZDRFRIVRMH
|
9.9 | IC50 | 4 | — | |
WWFBADABYQJEOH
|
9.9 | IC50 | 4 | — | |
PLYWKYGTXVRZIM
|
9.9 | IC50 | 4 | — | |
POHULTIMHMVEHW
|
9.9 | IC50 | 4 | — | |
RJFSUXPNRYMHRA
|
9.9 | IC50 | 4 | — | |
RZOMAMNKJPYXFW
|
9.9 | IC50 | 4 | — | |
USMNMZULIAYFEJ
|
9.9 | IC50 | 4 | — | |
BFDZAXLYGMAZBQ
|
9.9 | IC50 | 4 | — | |
CQVYWECRQQVMBR
|
9.9 | IC50 | 4 | — |