Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UZDRIDPZPMGZOL
|
8.8 | IC50 | 4 | — | |
BDMQXBKLHZGXQI
|
8.8 | IC50 | 4 | — | |
QDKKWLLPLUZTAW
|
8.8 | IC50 | 4 | — | |
VEXYMHUJQMBNMQ
|
8.8 | IC50 | 4 | — | |
DTQKHGKMBOLYLT
|
8.8 | IC50 | 4 | — | |
JMROEGRSMUVZFK
|
8.8 | IC50 | 4 | — | |
CJRRJWJKRXTHEF
|
8.7 | IC50 | 4 | — | |
SSSFMTDTKCJFRF
|
8.7 | IC50 | 4 | — | |
UTQRORGNZQVVQY
|
8.7 | IC50 | 4 | — | |
HMLMVOVUUWOJIT
|
8.7 | IC50 | 4 | — | |
KCGYMVKIHZQNLT
|
8.6 | IC50 | 4 | — | |
UILYFIYTPKDRTG
|
8.6 | IC50 | 4 | — | |
IMWXDQXYXIFOOQ
|
8.6 | IC50 | 4 | — | |
MWPLZFTURBIIPM
|
8.6 | IC50 | 4 | — | |
GWPDAIVBRKEDSC
|
8.6 | IC50 | 4 | — | |
ZVAPKOHBUPNLTN
|
8.5 | IC50 | 4 | — | |
XOQHYOIVBAXCRE
|
8.5 | IC50 | 4 | — | |
JZQVOGXMDSVEHZ
|
8.4 | IC50 | 4 | — | |
YILDOMMNMQFAPF
|
8.4 | IC50 | 4 | — | |
GQESRYREZHSCIP
|
8.4 | IC50 | 4 | — | |
WSCJOGHPXCRZQP
|
8.4 | IC50 | 4 | — | |
PZZILJUFSUVPJQ
|
8.3 | IC50 | 4 | — | |
RFCNFEVBCWVNCO
|
8.3 | IC50 | 4 | — | |
VWVDGIQYCWDZFS
|
8.3 | IC50 | 4 | — | |
QFUBXMRURPXZGY
|
8.2 | IC50 | 4 | — | |
JWVIACWDXBAAGB
|
8.2 | IC50 | 4 | — | |
MYMXIQGNYLCFBL
|
8.2 | IC50 | 4 | — | |
RHVHJNVUWWXGLK
|
8.2 | IC50 | 4 | — | |
GOJNRTLSOOOVJM
|
8.2 | IC50 | 4 | — | |
OUKQBVXVFXQAKN
|
8.1 | IC50 | 4 | — | |
GBNKXRKFDOPWQQ
|
8.0 | IC50 | 4 | — | |
NZHSSFSFHRZHMS
|
7.9 | IC50 | 3 | — | |
UMNPTGPXWSXOOY
|
7.9 | IC50 | 4 | — | |
AHMBFQAMCZCYCG
|
7.6 | IC50 | 4 | — | |
PGWUOFRMVJEOIN
|
7.6 | IC50 | 3 | — |