Target Details
| UniProt AC | Q2QC95 |
|---|---|
| Gene Symbol | blaoxa-10 |
| Protein Name | Beta-lactamase |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00905 (Transpeptidase) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 9.56
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RQPNOZBYGYYABS
|
10.4 | IC50 | 4 | — | |
UMHFRIKKMWUBNA
|
10.3 | IC50 | 4 | — | |
ABGWLUMGGAKQLX
|
10.3 | IC50 | 4 | — | |
HCBQCTAFMHAHIT
|
10.3 | IC50 | 4 | — | |
VQFVDKZCXCUSNA
|
10.3 | IC50 | 4 | — | |
ABAPJYDJVJVZSN
|
10.3 | IC50 | 4 | — | |
BWZLKGTWPNUCTO
|
10.3 | IC50 | 4 | — | |
CQDLIMUHAKMXNT
|
10.3 | IC50 | 4 | — | |
BGVFFBGEJPULGP
|
10.3 | IC50 | 4 | — | |
PPVAWQLUAZOCPF
|
10.2 | IC50 | 4 | — | |
QHJWADHROHWYDE
|
10.2 | IC50 | 4 | — | |
MMDRDTANGPSQJU
|
10.2 | IC50 | 4 | — | |
XXMRXEKEKMQIKH
|
10.2 | IC50 | 4 | — | |
IDKMTIOFCUCPGQ
|
10.2 | IC50 | 4 | — | |
QMKPKGKQGOYUFS
|
10.2 | IC50 | 3 | — | |
FEUZVDVCIDGGHY
|
10.1 | IC50 | 4 | — | |
LHGHDVNQBZMSRJ
|
10.1 | IC50 | 4 | — | |
VUYNFVVRABLCCA
|
10.1 | IC50 | 4 | — | |
JALKVYMRKKEWJK
|
10.1 | IC50 | 4 | — | |
XJPGGPKEFJDYDK
|
10.1 | IC50 | 4 | — | |
AYVVPNLUKSCPMU
|
10.1 | IC50 | 4 | — | |
NNFCNZSFFWFISR
|
10.1 | IC50 | 4 | — | |
PSUWTYNLWBIWIE
|
10.1 | IC50 | 4 | — | |
RXRGCIXNNYNDOB
|
10.1 | IC50 | 4 | — | |
XFHGATVLSRCKLK
|
10.1 | IC50 | 4 | — | |
AUYJNPQTWCJSFY
|
10.1 | IC50 | 4 | — | |
BFOYHAUOQCJINB
|
10.1 | IC50 | 4 | — | |
CAPREPJCVIJSJF
|
10.1 | IC50 | 4 | — | |
CRWZLJNNDOWHSX
|
10.0 | IC50 | 4 | — | |
DALYKNCYQQMDQU
|
10.0 | IC50 | 4 | — | |
GZBHDBFPVJZAKJ
|
10.0 | IC50 | 4 | — | |
RXRGCIXNNYNDOB
|
10.0 | IC50 | 4 | — | |
ADGAXIHGUNIVHL
|
10.0 | IC50 | 4 | — | |
ZUMVYUASFRNBGF
|
10.0 | IC50 | 4 | — | |
AWFLVGLEZADZME
|
10.0 | IC50 | 4 | — | |
FXAAYEGOAOZVQG
|
10.0 | IC50 | 4 | — | |
NGJUIXRTMZQSAK
|
10.0 | IC50 | 4 | — | |
ZYNDVCSMOHTMPY
|
10.0 | IC50 | 3 | — | |
BKJNWVSHORBYDI
|
10.0 | IC50 | 4 | — | |
SJTLDCMGGRCPJQ
|
10.0 | IC50 | 3 | — | |
WGCIOOTXJABATI
|
10.0 | IC50 | 4 | — | |
CLEQRMCQLNNGRY
|
10.0 | IC50 | 4 | — | |
LZEADKZZIQVDOZ
|
10.0 | IC50 | 4 | — | |
OQTUJIHTSYMXJD
|
10.0 | IC50 | 4 | — | |
PPVAWQLUAZOCPF
|
10.0 | IC50 | 4 | — | |
UNWJCMBQRPPTIH
|
10.0 | IC50 | 4 | — | |
FXAAYEGOAOZVQG
|
10.0 | IC50 | 4 | — | |
KIHWPFSYAMCZDY
|
10.0 | IC50 | 4 | — | |
NJKDZCGDZKEPQP
|
10.0 | IC50 | 4 | — | |
OGSYXYCAUVSMCS
|
10.0 | IC50 | 3 | — |