Target Details
| UniProt AC | Q2M2I8 |
|---|---|
| Gene Symbol | AAK1 |
| Protein Name | AP2-associated protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 98
- Clinical molecules 15
- Avg pChEMBL 7.62
Active Molecules (98)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CJIAUJUVHMAHQC
|
7.4 | Ki | 4 | — | |
YLVDJOXELSCRPM
|
7.4 | IC50 | 3 | — | |
HWXVIOGONBBTBY
|
7.4 | Kd | 27 | — | |
BPNUQXPIQBZCMR
|
7.4 | Kd | 83 | Yes | |
MCYCSSJHDPRHBZ
|
7.4 | Ki | 4 | — | |
BMGQWWVMWDBQGC
|
7.3 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.3 | Kd | 91 | Yes | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
IAYGCINLNONXHY
|
7.3 | Kd | 50 | — | |
NKCMEGZSWOVKIL
|
7.3 | IC50 | 3 | — | |
SENOTLIGBLGKGP
|
7.3 | IC50 | 3 | — | |
JTSLALYXYSRPGW
|
7.2 | Kd | 8 | — | |
KMVVQXBUHOYQKZ
|
7.2 | Ki | 3 | — | |
XZXHXSATPCNXJR
|
7.2 | Kd | 165 | Yes | |
CTNPALGJUAXMMC
|
7.2 | Kd | 151 | — | |
OEZHSZIDGUKBRK
|
7.1 | IC50 | 10 | — | |
RDROKTFULACVDQ
|
7.1 | IC50 | 8 | — | |
JEESDCKVMQTTMP
|
7.0 | IC50 | 3 | — | |
MXOVNNMQDFPQKY
|
7.0 | IC50 | 3 | — | |
UZWDCWONPYILKI
|
7.0 | Kd | 47 | — | |
CHQYAWLKOUOTQO
|
7.0 | IC50 | 20 | — | |
JNYMSOJGKCXZLV
|
7.0 | IC50 | 3 | — | |
HFNKQEVNSGCOJV
|
6.9 | Kd | 65 | — | |
JTVBXQAYBIJXRP
|
6.9 | Kd | 20 | — | |
ALKJNCZNEOTEMP
|
6.9 | Kd | 55 | — | |
PIQCTGMSNWUMAF
|
6.8 | Kd | 137 | Yes | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
KDKUVYLMPJIGKA
|
6.7 | Kd | 91 | Yes | |
MENVSADYTLLXLP
|
6.7 | IC50 | 6 | — | |
ODOJVROSIRINJT
|
6.7 | IC50 | 3 | — | |
IYHHRZBKXXKDDY
|
6.7 | IC50 | 6 | — | |
WJRRGYBTGDJBFX
|
6.6 | Kd | 16 | Yes | |
RXQXACYMRVINQU
|
6.5 | IC50 | 5 | — | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
OYONTEXKYJZFHA
|
6.5 | Kd | 69 | Yes | |
QVADIDYLQUXJQI
|
6.5 | IC50 | 2 | — | |
PKEYNQACQWYICF
|
6.4 | IC50 | 6 | — | |
RZUOCXOYPYGSKL
|
6.4 | Kd | 8 | — | |
NHHQJBCNYHBUSI
|
6.4 | Kd | 220 | — | |
BMWMKGNVAMXXCH
|
6.4 | Kd | 6 | — | |
FVMPOTYRHZJMAJ
|
6.4 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.3 | Kd | 231 | Yes | |
GUBJNPWVIUFSTR
|
6.3 | Kd | 103 | — | |
PBCZSGKMGDDXIJ
|
6.2 | Kd | 68 | Yes | |
UJIAQDJKSXQLIT
|
6.1 | Kd | 38 | — | |
ZCBUQCWBWNUWSU
|
6.0 | Kd | 59 | — | |
ZZSBPGIGIUFJRA
|
6.0 | Kd | 46 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |