Target Details
| UniProt AC | Q2M2I8 |
|---|---|
| Gene Symbol | AAK1 |
| Protein Name | AP2-associated protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 98
- Clinical molecules 15
- Avg pChEMBL 7.62
Active Molecules (98)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSZZLVNYBNWVDL
|
9.3 | IC50 | 2 | — | |
LAHYYLXFCBPDDW
|
9.3 | IC50 | 2 | — | |
NGBWQVJCOYTGOR
|
9.3 | IC50 | 8 | — | |
RKBMAROJKLHAMI
|
9.3 | IC50 | 6 | — | |
QHPJIUARPKBLQQ
|
9.2 | IC50 | 3 | — | |
UJFBQMHGCCSHRP
|
9.2 | IC50 | 2 | — | |
ZVSNSFQQKSZZMY
|
9.2 | IC50 | 7 | — | |
IZPCBCVMTALJQY
|
9.1 | IC50 | 3 | — | |
KPYMRFGAAXFXIK
|
9.1 | IC50 | 2 | — | |
MDBWZAGCBGPXST
|
9.1 | IC50 | 2 | — | |
HDBIRBUHIXXLDF
|
9.0 | IC50 | 4 | — | |
SVNVPNHWFJFRLZ
|
9.0 | IC50 | 8 | — | |
HINOQCZIDBNXEI
|
9.0 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
8.9 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
8.9 | Kd | 213 | — | |
HVHRHDHQHUAOQI
|
8.9 | IC50 | 5 | — | |
PFMMJDPMFCVRCB
|
8.9 | IC50 | 4 | — | |
FFTUIKFDUYMWTI
|
8.8 | IC50 | 5 | — | |
YFNWWNRZJGMDBR
|
8.7 | Kd | 35 | — | |
RKAHOQATMSONTM
|
8.7 | IC50 | 6 | — | |
ZFXGOGALEGXWEL
|
8.6 | IC50 | 5 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
GOOYSJIWTIHOGW
|
8.5 | IC50 | 3 | — | |
XYXJLVVKIBEGES
|
8.5 | IC50 | 2 | — | |
KOZFSFOOLUUIGY
|
8.3 | Kd | 88 | Yes | |
OSVUGUHRKMMBSE
|
8.3 | Kd | 170 | — | |
FMNWOBLAZAYOSG
|
8.2 | IC50 | 5 | — | |
NXSJMRCTGYTSTK
|
8.2 | Kd | 200 | — | |
USXZHEGWWNBLBI
|
8.2 | Ki | 4 | — | |
YKGQUBOYHDWACY
|
8.2 | IC50 | 2 | — | |
XUZMWHLSFXCVMG
|
8.1 | Kd | 24 | — | |
CGXOKVWAHQLXGW
|
8.1 | IC50 | 2 | — | |
RYYNGWLOYLRZLK
|
8.1 | Kd | 45 | — | |
AKUJIVTZSHCXRK
|
8.0 | IC50 | 2 | — | |
GXQWWDBZTZLIAJ
|
8.0 | Ki | 3 | — | |
WINHZLLDWRZWRT
|
8.0 | Kd | 201 | Yes | |
GCTFTMWXZFLTRR
|
7.9 | IC50 | 7 | — | |
IPEXHQGMTHOKQV
|
7.9 | Kd | 12 | — | |
UCBIQZUJJSVQHL
|
7.8 | IC50 | 8 | — | |
LOLPPWBBNUVNQZ
|
7.8 | Kd | 97 | Yes | |
YSMDVXCUNQWGNN
|
7.7 | Ki | 4 | — | |
DPCPNRYPXUUJCP
|
7.7 | Ki | 4 | — | |
XLSYZSRXVVCHLS
|
7.7 | Kd | 48 | — | |
IIKPYJZUOZRTIB
|
7.5 | Ki | 4 | — | |
HJDMEPOCEJXNJU
|
7.5 | IC50 | 3 | — | |
NTOMZGNNDKIPEH
|
7.5 | Ki | 4 | — | |
INTMVZKGQXMUML
|
7.5 | Ki | 3 | — | |
JOOXLOJCABQBSG
|
7.5 | Kd | 139 | — | |
KRIUNPBAQZGFQA
|
7.5 | Kd | 76 | — | |
QDITZBLZQQZVEE
|
7.5 | Kd | 19 | — |