Target Details
| UniProt AC | Q2FYS5 |
|---|---|
| Gene Symbol | parE |
| Protein Name | DNA topoisomerase 4 subunit B |
| Organism | Staphylococcus aureus (strain NCTC 8325 / PS 47) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 4
- Clinical molecules 0
- Avg pChEMBL 6.91
Active Molecules (4)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWGVZRSKDSKOCX
|
7.8 | IC50 | 3 | — | |
RPPRAYQNSDDYNW
|
7.6 | IC50 | 2 | — | |
RXPOVSSVBGRCOL
|
6.2 | IC50 | 2 | — | |
ZFMCWMJGTDHLKI
|
6.0 | IC50 | 2 | — |