Target Details
| UniProt AC | Q27552 |
|---|---|
| Gene Symbol | DHFR-TS |
| Protein Name | Bifunctional dihydrofolate reductase-thymidylate synthase |
| Organism | Cryptosporidium parvum |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) PF00303 (Thymidylat_synt) |
Summary
- Multi-target molecules 20
- Clinical molecules 0
- Avg pChEMBL 7.77
Active Molecules (20)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JPENSYBRTSIYGO
|
9.0 | IC50 | 3 | — | |
JPENSYBRTSIYGO
|
8.7 | IC50 | 5 | — | |
USMIUYUTXWJTSL
|
8.7 | IC50 | 3 | — | |
XZXVRKHUCSXVBM
|
8.7 | IC50 | 3 | — | |
KEPKKUKRTDFXHZ
|
8.2 | IC50 | 2 | — | |
NUZPENCTXJLJCY
|
8.1 | IC50 | 2 | — | |
VOTVRUAOKKCDKI
|
8.0 | IC50 | 2 | — | |
NQBNSJKYKJECKP
|
7.8 | IC50 | 2 | — | |
DATCFVVEPPDLRQ
|
7.7 | IC50 | 3 | — | |
DATCFVVEPPDLRQ
|
7.7 | IC50 | 3 | — | |
YYCPXVRHQUEVAW
|
7.7 | IC50 | 2 | — | |
UKKLVFSCEPWYNJ
|
7.6 | IC50 | 2 | — | |
JPENSYBRTSIYGO
|
7.5 | IC50 | 2 | — | |
GWGFEUVZNZOACY
|
7.4 | IC50 | 2 | — | |
KZCLZTHWXHXZDO
|
7.4 | IC50 | 2 | — | |
LFVCHCWJLBIVBU
|
7.2 | IC50 | 2 | — | |
JYPKSMDSADPSKN
|
7.1 | IC50 | 2 | — | |
RUQVXLIOJPKNCM
|
7.1 | IC50 | 3 | — | |
VDHBMZRBPMTLGE
|
6.9 | IC50 | 2 | — | |
RUQVXLIOJPKNCM
|
6.8 | IC50 | 4 | — |