Target Details
| UniProt AC | Q16832 |
|---|---|
| Gene Symbol | DDR2 |
| Protein Name | Discoidin domain-containing receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 233
- Clinical molecules 21
- Avg pChEMBL 7.22
Associated Diseases (1)
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBPYILGKFZZVDX
|
6.8 | Kd | 130 | Yes | |
PBHDCPWPSOSGGD
|
6.8 | IC50 | 2 | — | |
CTQCFMSNNVNUQZ
|
6.8 | IC50 | 2 | — | |
NHCXDULQCCCWLO
|
6.8 | IC50 | 3 | — | |
ZCWXCBKGPJOAFQ
|
6.8 | IC50 | 13 | — | |
NYVPWRKNAAFYQA
|
6.8 | IC50 | 2 | — | |
WAJTXTQMISPZDI
|
6.8 | Ki | 2 | — | |
DKNUPRMJNUQNHR
|
6.7 | Kd | 33 | — | |
GNDBDDNLWIOKDN
|
6.7 | IC50 | 5 | — | |
RYCUVZMYBSSMAE
|
6.7 | IC50 | 2 | — | |
CMJJZRAAQMUAFH
|
6.7 | IC50 | 9 | — | |
FAYAUAZLLLJJGH
|
6.7 | IC50 | 36 | Yes | |
WWIJZOWOWLGRSG
|
6.7 | IC50 | 2 | — | |
DRNRCLNUHIQXOJ
|
6.7 | IC50 | 4 | — | |
RALKOVHFGYUBAB
|
6.7 | IC50 | 5 | — | |
FXUBVXGXYWZNJY
|
6.7 | IC50 | 2 | — | |
WOSKHXYHFSIKNG
|
6.7 | Kd | 24 | — | |
XEKBRFPQVSQWMU
|
6.7 | IC50 | 3 | — | |
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
VWMJHAFYPMOMGF
|
6.6 | Kd | 15 | — | |
DDPFCUXJEFSBMK
|
6.6 | IC50 | 2 | — | |
MWFIUFYSLJRFQM
|
6.6 | IC50 | 2 | — | |
RZOMPFGUSZPJBC
|
6.5 | IC50 | 3 | — | |
XVBSTEJSDUMWMA
|
6.5 | IC50 | 3 | — | |
AIKGYQDFIJRQIY
|
6.5 | IC50 | 9 | — | |
FTDWSWREBGYXDZ
|
6.5 | IC50 | 10 | — | |
HJWMLCDGRWWLAQ
|
6.5 | IC50 | 3 | — | |
IVUGFMLRJOCGAS
|
6.5 | Kd | 9 | — | |
MWKSRKSEWLRPBL
|
6.5 | Kd | 1075 | — | |
YLNAPFRQMKNPTD
|
6.5 | Ki | 2 | — | |
GMHKDZXPTJDOJO
|
6.5 | IC50 | 2 | — | |
BGQOUQWQPRPBKN
|
6.5 | IC50 | 7 | — | |
DQHVUKLVCBJBLM
|
6.5 | IC50 | 8 | — | |
RHSMFYIHIIADSH
|
6.5 | IC50 | 5 | — | |
UHTHHESEBZOYNR
|
6.5 | Kd | 66 | Yes | |
IKENQUDOTQBCJH
|
6.5 | IC50 | 18 | — | |
PGNPRFGVXQKJFG
|
6.5 | IC50 | 4 | — | |
GYFKBVBCLVBDJM
|
6.4 | IC50 | 2 | — | |
IQMKTZJMVCUBEI
|
6.4 | Kd | 2 | — | |
QUOWKTGPIJLRIN
|
6.4 | Kd | 2 | — | |
UIARLYUEJFELEN
|
6.4 | Kd | 289 | Yes | |
XWIZEHJOUXPUMM
|
6.4 | Kd | 2 | — | |
AOZPVMOOEJAZGK
|
6.4 | IC50 | 2 | — | |
FNHKPVJBJVTLMP
|
6.4 | Kd | 29 | — | |
HXHAJRMTJXHJJZ
|
6.4 | IC50 | 52 | Yes | |
ZCCPLJOKGAACRT
|
6.4 | Kd | 599 | — | |
CMJJZRAAQMUAFH
|
6.4 | IC50 | 2 | — | |
IZGJBYFGTKCESG
|
6.3 | IC50 | 2 | — | |
OPEMWSXQLXWPSB
|
6.3 | IC50 | 2 | — | |
DIMLYBUSJYNUFT
|
6.3 | IC50 | 6 | — |