Target Details
| UniProt AC | Q16832 |
|---|---|
| Gene Symbol | DDR2 |
| Protein Name | Discoidin domain-containing receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 233
- Clinical molecules 21
- Avg pChEMBL 7.22
Associated Diseases (1)
Active Molecules (233)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CYYRPFWAMVGRGT
|
7.3 | IC50 | 3 | — | |
CTZOFTNYJRGNGO
|
7.3 | IC50 | 3 | — | |
XXJWYDDUDKYVKI
|
7.3 | Kd | 52 | — | |
ZGBAJMQHJDFTQJ
|
7.3 | Kd | 15 | — | |
SDYGMEWQBSWSIW
|
7.3 | IC50 | 6 | — | |
HYWXBDQAYLPMIX
|
7.3 | IC50 | 3 | Yes | |
WPXVVAWAHQHJPF
|
7.3 | IC50 | 41 | — | |
GZOONDJISKPFEJ
|
7.2 | IC50 | 4 | — | |
BPQBMWJXOIQOCG
|
7.2 | IC50 | 3 | — | |
BCIITSAFUJGIEG
|
7.2 | IC50 | 3 | — | |
SKDBXDGKLQALIZ
|
7.2 | IC50 | 15 | — | |
DZVQBRGQNWDWIG
|
7.2 | IC50 | 6 | — | |
MOONEVNPHKFNGV
|
7.2 | Kd | 4 | — | |
KZVIZFHCMVWFNT
|
7.2 | IC50 | 7 | — | |
VNBRGSXVFBYQNN
|
7.2 | Kd | 22 | Yes | |
YHVHYWYQEFELOW
|
7.2 | IC50 | 44 | — | |
RIWKVLUOTMXONS
|
7.2 | IC50 | 5 | — | |
OTKXMYZOSPIKMY
|
7.1 | IC50 | 3 | — | |
VAPRWSMRTJIVDQ
|
7.1 | IC50 | 4 | — | |
LAXWYKGMTZIWKO
|
7.1 | IC50 | 3 | — | |
LQSGDXCDNZWTJN
|
7.1 | IC50 | 17 | — | |
UEHGHDJPDQDZPX
|
7.1 | IC50 | 3 | — | |
QTYVZNNBMDNHJL
|
7.1 | IC50 | 3 | — | |
SERAEYFDVQXTIX
|
7.1 | Kd | 2 | — | |
PHXJVRSECIGDHY
|
7.1 | Kd | 59 | — | |
SHPFDGWALWEPGS
|
7.1 | Kd | 35 | — | |
CUDVHEFYRIWYQD
|
7.0 | Kd | 11 | — | |
GYBZVTMKISJGBF
|
7.0 | IC50 | 3 | — | |
RFEWCQAWLXXDQI
|
7.0 | IC50 | 5 | — | |
XQZFAZMTCODCDH
|
7.0 | IC50 | 3 | — | |
CUIHSIWYWATEQL
|
7.0 | Kd | 61 | Yes | |
GUBJNPWVIUFSTR
|
7.0 | Kd | 103 | — | |
MXYXKUBTRKHYAM
|
7.0 | IC50 | 3 | — | |
RKDBIDWPRDZSFA
|
7.0 | IC50 | 2 | — | |
CKFSGFBIQDUWKV
|
7.0 | IC50 | 5 | — | |
DDLPXZXBWGJRGK
|
7.0 | IC50 | 4 | — | |
ZHAGZTJIWAFRBI
|
7.0 | IC50 | 3 | — | |
APPXQUDJLJXULP
|
6.9 | IC50 | 47 | — | |
UYAJMVJVPHCOJN
|
6.9 | IC50 | 3 | — | |
UXXQOJXBIDBUAC
|
6.9 | Kd | 21 | Yes | |
XTFQLAOUVSZDDX
|
6.9 | IC50 | 3 | — | |
DNMQPIQPJLMWPY
|
6.9 | IC50 | 3 | — | |
HKHQEYYGONFDJK
|
6.9 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
6.9 | IC50 | 92 | — | |
BNRXMSGHPVYSDK
|
6.9 | IC50 | 24 | — | |
CAWFLWKFZFPVQV
|
6.9 | IC50 | 3 | — | |
UHWZHRQDJOKBQY
|
6.9 | IC50 | 3 | — | |
KYENXKDRIQKRJP
|
6.9 | IC50 | 5 | — | |
JUUFLLKHNYWHKP
|
6.9 | Kd | 12 | — | |
KTUFNOKKBVMGRW
|
6.8 | Kd | 38 | Yes |